SCHEMBL7149480

SCHEMBL7149480

CC1(C)CCC(C)(C)c2cc(C(=O)O)c(O)cc21

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 19/20 0.69
RARB P10826 7/20 0.65
RARG P13631 7/20 0.57
RARA P10276 4/20 0.57
RXRB P28702 5/20 0.53
RXRG P48443 5/20 0.53
MEN1 O00255 1/20 0.50
CYP26A1 O43174 1/20 0.50
ABCB11 O95342 1/20 0.50
ESR1 P03372 1/20 0.50
PGR P06401 1/20 0.50
HTR1A P08908 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CHRM1 P11229 1/20 0.50
DRD1 P21728 1/20 0.50
TBXA2R P21731 1/20 0.50
SLC6A2 P23975 1/20 0.50
ADRA1A P35348 1/20 0.50
OPRM1 P35372 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30701833 1.00 RXRA (0.69) RXRARARBRARGRARARXRB
SCHEMBL28646163 0.88 RXRA (0.59) RXRARARBRARGRARARXRB
SCHEMBL726366 0.85 RXRA (0.59) RXRARARBRARGRARARXRB
SCHEMBL1073920 0.82 RXRA (1.00) RXRARARBRARGRARARXRB
SCHEMBL5359740 0.81 RXRA (0.71) RXRARARBRARGRARARXRB
SCHEMBL2191766 0.80 RXRA (0.55) RXRARARBRARGRARARXRB
SCHEMBL2196140 0.80 RXRA (0.55) RXRARARBRARGRARARXRB
SCHEMBL2196986 0.80 RXRA (0.55) RXRARARBRARGRARARXRB
SCHEMBL2193183 0.80 RXRA (0.81) RXRARARBRARGRARARXRB
SCHEMBL6889176 0.80 RXRA (1.00) RXRARARBRARGRARARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240246900-A1 SYNTHESIS OF TETRAHYDRONAPHTHALENOLS AND USES THEREOF Io Therapeutics, Inc. 2024-07-25 US disclosed
US-11976021-B2 Synthesis of tetrahydronaphthalenols and uses thereof Io Therapeutics, Inc. (US) 2024-05-07 US disclosed
WO-2024006732-A1 SYNTHESIS OF TETRAHYDRONAPHTHALENOLS AND USES THEREOF Io Therapeutics, Inc. (US) 2024-01-04 WO disclosed
US-20230416190-A1 SYNTHESIS OF TETRAHYDRONAPHTHALENOLS AND USES THEREOF Io Therapeutics, Inc. 2023-12-28 US disclosed
US-8765719-B2 Therapeutic drug for adult T-cell leukemia KAGOSHIMA UNIVERSITY (JP) 2014-07-01 US disclosed
US-8765719-B2 Therapeutic drug for adult T-cell leukemia KAGOSHIMA UNIVERSITY (JP) 2014-07-01 US disclosed
EP-2345409-A1 THERAPEUTIC AGENT FOR ADULT T-CELL LEUKEMIA Kagoshima University (JP) 2011-07-20 EP disclosed
US-20110172185-A1 THERAPEUTIC DRUG FOR ADULT T-CELL LEUKEMIA KAGOSHIMA UNIVERSITY (JP) 2011-07-14 US disclosed
US-20110172185-A1 THERAPEUTIC DRUG FOR ADULT T-CELL LEUKEMIA KAGOSHIMA UNIVERSITY (JP) 2011-07-14 US disclosed
US-6610744-B2 Administering to a mammal a retinoid campound which binds specifically or selectively to a RAR alpha retinoid receptors in preference over RAR beta and RAR Gamma retinoid receptors, for therapy and prophylaxisof disease or condition ALLERGAN, INC. 2003-08-26 US disclosed
US-20020077360-A1 Methods of treatment with compounds having RAR alpha receptor specific or selective activity ALLERGAN SALES, INC. 2002-06-20 US disclosed
US-6342602-B1 BIND SPECIFICALLY OR SELECTIVELY TO RAR-ALPHA RECEPTORS ALLERGAN SALES, INC. 2002-01-29 US disclosed
EP-0876330-B1 ARYL OR HETEROARYL AMIDES OF TETRAHYDRONAPHTHALENE, CHROMAN, THIOCHROMAN AND 1,2,3,4-TETRAHYDROQUINOLINE CARBOXYLIC ACIDS HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES INC (US) 2001-03-28 EP disclosed
US-6124455-A Aryl or heteroaryl amides of tetrahydronaphthalene, chroman, thiochroman and 1,2,3,4-tetrahydroquinoline carboxylic acids, having an electron withdrawing substituent in the aromatic or heteroaromatic moiety, having retinoid-like biological activity ALLERGAN SALES, INC. (US) 2000-09-26 US disclosed
US-6034244-A ANTIINFLAMMATORY AGENTS; SKIN DISORDERS; ANTICANCER AGENT ALLERGAN SALES, INC. (US) 2000-03-07 US disclosed
US-5965606-A RETINOID RECEPTORS, 2-FLUORO-4-(2',2',4',4'-TETRAMETHYL-8'-TRIFLUOROMETHYLCHROMAN-6' -YL)CARBAMOYL BENZOIC ACID FOR TREATING MONOCYTIC LEUKEMIA ALLERGAN SALES, INC. (US) 1999-10-12 US disclosed
US-5856490-A Aryl or heteroaryl amides of tetrahydronaphthalene, chroman, thiochroman and 1,2,3,4-tetrahydroquinoline carboxylic acids, having an electron withdrawing substituent in the aromatic or heteroaromatic moiety, having retinoid-like biological activity ALLERGAN (US) 1999-01-05 US disclosed
EP-0869782-A2 METHODS OF TREATMENT WITH COMPOUNDS HAVING RAR $g(a)? RECEPTOR SPECIFIC OR SELECTIVE ACTIVITY Vision Pharmaceuticals L.P. (US) 1998-10-14 EP disclosed
US-5675024-A RETINOID RECEPTOR AGONISTS ALLERGAN (US) 1997-10-07 US disclosed
WO-1997024116-A2 METHODS OF TREATMENT WITH COMPOUNDS HAVING RARα RECEPTOR SPECIFIC OR SELECTIVE ACTIVITY VISION PHARMACEUTICALS L.P. (US) 1997-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020077360-A1 Methods of treatment with compounds having RAR alpha receptor specific or selective activity RARG, RARA, RARB RXRA 5/4885RARB 3/4885RARG 1/4885
US-20240246900-A1 SYNTHESIS OF TETRAHYDRONAPHTHALENOLS AND USES THEREOF DHPS, LSS, CYP8B1 RXRA 968/4885RARB 1499/4885RARG 932/4885
US-20110172185-A1 THERAPEUTIC DRUG FOR ADULT T-CELL LEUKEMIA CBR3, CD47, ATL3 RXRA 1135/4885RARB 2945/4885RARG 2656/4885
US-11976021-B2 Synthesis of tetrahydronaphthalenols and uses thereof DHPS, LSS, CYP8B1 RXRA 968/4885RARB 1499/4885RARG 932/4885
US-20230416190-A1 SYNTHESIS OF TETRAHYDRONAPHTHALENOLS AND USES THEREOF DHPS, LSS, CYP8B1 RXRA 968/4885RARB 1499/4885RARG 932/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.