SCHEMBL7154383

SCHEMBL7154383

CSc1ccccc1-c1cc(C)oc(=O)c1-c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
RAB9A P51151 3/20 0.39
HPGD P15428 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
USP2 O75604 1/20 0.38
USP1 O94782 1/20 0.38
USP8 P40818 1/20 0.38
OTUB1 Q96FW1 1/20 0.38
USP36 Q9P275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7154393 0.82 MAOA (0.42) MAOAMAOBRAB9ANPC1ACLY
SCHEMBL7108266 0.80 PTGS2 (0.45) MAOAMAOBLMNAUSP2USP1
SCHEMBL5709000 0.74 PTGS2 (0.59)
SCHEMBL7024957 0.68 PTGS2 (0.49)
SCHEMBL7154386 0.65 MAOA (0.38) MAOAMAOBALDH1A1MAPTRAB9A
SCHEMBL7372656 0.64 ALOX5 (0.50) ALDH1A1KDM4EMAPTRAB9AHPGD
SCHEMBL7374057 0.63 NPY5R (0.39) ALDH1A1KDM4EMAPTRAB9AHPGD
SCHEMBL5890646 0.62 KDM4E (0.52) ALDH1A1KDM4EMAPTRAB9AHPGD
SCHEMBL3480552 0.62 CYP2A6 (0.54) ALDH1A1KDM4EMAPTRAB9AHPGD
SCHEMBL31087243 0.62 KDM4E (0.52) ALDH1A1KDM4EMAPTRAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299372-A1 PYRONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 2003-04-09 EP disclosed
WO-2002002547-A1 PYRONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 2002-01-10 WO disclosed