SCHEMBL7154393

SCHEMBL7154393

CSc1ccc(-c2cc(C)oc(=O)c2-c2cccnc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
CYP19A1 P11511 1/20 0.38
ACLY P53396 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ELANE P08246 1/20 0.37
PTGS2 P35354 1/20 0.37
CYP2A6 P11509 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024957 0.84 PTGS2 (0.49) PTGS2
SCHEMBL5709000 0.82 PTGS2 (0.59) PTGS2
SCHEMBL7154383 0.82 MAOA (0.41) MAOAMAOBACLYNPC1RAB9A
SCHEMBL7022294 0.79 PTGS2 (0.45) PTGS2
SCHEMBL7029451 0.78 PTGS1 (0.43) PTGS2
SCHEMBL7259908 0.75 PTGS2 (0.46) RAB9APTGS2
SCHEMBL7108266 0.74 PTGS2 (0.45) MAOAMAOBACLYPTGS2
SCHEMBL7154386 0.73 MAOA (0.38) MAOAMAOBACLYNPC1RAB9A
SCHEMBL7028615 0.72 RAB9A (0.41) MAOBRAB9APTGS2
SCHEMBL8423037 0.71 PTGS2 (0.51) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299372-A1 PYRONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 2003-04-09 EP disclosed
WO-2002002547-A1 PYRONES AS INHIBITORS OF CYCLOOXYGENASE-2 MERCK FROSST CANADA & CO. (CA) 2002-01-10 WO disclosed