SCHEMBL7160977

SCHEMBL7160977

Nc1cc2c(cc1Sc1ccc(F)cc1F)C(=O)CC2

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.62
PTGS1 P23219 2/20 0.62
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
HSD17B10 Q99714 1/20 0.40
HSD17B1 P14061 1/20 0.36
SRD5A1 P18405 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK14 Q16539 1/20 0.34
PBRM1 Q86U86 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13178557 0.78 PTGS2 (0.53) PTGS2PTGS1CASP1CASP7HSD17B10
Ethylene SCHEMBL7162487 0.78 PTGS2 (0.55) PTGS2PTGS1ALDH1A1
SCHEMBL29385521 0.77 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL2464202 0.77 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL10942403 0.73 PTGS2 (0.62) PTGS2PTGS1CASP1CASP7HSD17B10
SCHEMBL30957305 0.72 CASP1 (0.50) PTGS2PTGS1CASP1CASP7HSD17B10
SCHEMBL21505155 0.72 CASP1 (0.50) PTGS2PTGS1CASP1CASP7HSD17B10
SCHEMBL11181698 0.70 CASP1 (0.45) PTGS2CASP1CASP7HSD17B10ALDH1A1
SCHEMBL576377 0.70 ALDH1A1 (0.46) PTGS2PTGS1ALDH1A1MAPK14
SCHEMBL30452220 0.70 ALDH1A1 (0.46) PTGS2PTGS1ALDH1A1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE38103-E1 5-methanesulfonamido-1-indanones as an inhibitor of cyclooxygenase-2 MERCK FROSST CANADA & CO. (CA) 2003-04-29 US disclosed
EP-0673366-B1 5-METHANESULFONAMIDO-1-INDANONES AS AN INHIBITOR OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC (CA) 1998-10-14 EP disclosed
US-5604260-A 5-methanesulfonamido-1-indanones as an inhibitor of cyclooxygenase-2 MERCK FROSST CANADA INC. (CA) 1997-02-18 US disclosed
EP-0673366-A1 5-METHANESULFONAMIDO-1-INDANONES AS AN INHIBITOR OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 1995-09-27 EP disclosed
WO-1994013635-A1 5-METHANESULFONAMIDO-1-INDANONES AS AN INHIBITOR OF CYCLOOXYGENASE-2 MERCK FROSST CANADA INC. (CA) 1994-06-23 WO disclosed