SCHEMBL7165451

SCHEMBL7165451

O=C(O)CC(=O)[N]c1cccnc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.47
PLOD2 O00469 1/20 0.45
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
ALDH1A1 P00352 2/20 0.43
APP P05067 1/20 0.43
GAA P10253 1/20 0.43
HCAR3 P49019 1/20 0.43
HCAR2 Q8TDS4 1/20 0.43
TBXAS1 P24557 8/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
USP2 O75604 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
NOS3 P29474 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5509513 0.81 NOS3 (0.47) NAPRTHTR3EHTR3BHTR3AHTR3D
SCHEMBL2229589 0.79 MAPT (0.41) ALDH1A1GAANPC1RAB9AMAPT
SCHEMBL1008978 0.74 HTR3E (0.60) NAPRTHTR3EHTR3BHTR3AHTR3D
SCHEMBL5509993 0.73 NOS3 (0.48) PLOD2HTR3EHTR3BHTR3AHTR3D
Malonic Acid SCHEMBL28183811 0.71 NAPRT (0.53) NAPRTPLOD2ALDH1A1APPGAA
SCHEMBL2694778 0.69 PLOD2 (0.79) NAPRTPLOD2ALDH1A1APPGAA
SCHEMBL7497348 0.69 HTR3E (0.45) NAPRTHTR3EHTR3BHTR3AHTR3D
SCHEMBL7168276 0.69 MEN1 (0.42) GAANPC1RAB9AMAPTHDAC1
SCHEMBL27582165 0.67 NAPRT (0.73) NAPRTTBXAS1
SCHEMBL307606 0.67 ALDH1A1 (0.71) ALDH1A1NPC1PKMRAB9AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-B1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2003-05-07 EP claimed