SCHEMBL7167229

SCHEMBL7167229

Cc1ccc(-c2ccc3c(c2)C=C(C(=O)NC2CCN(C4CCOCC4)CC2)CCO3)cc1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.55
CCR2 P41597 2/20 0.40
CCR7 P32248 1/20 0.40
CXCR3 P49682 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7221530 0.92 CCR5 (0.46) CCR5CXCR3
SCHEMBL7223524 0.88 CCR5 (0.53) CCR5
SCHEMBL7223533 0.87 CCR5 (0.54) CCR5CCR2
SCHEMBL7215850 0.87 CCR5 (0.55) CCR5
SCHEMBL7222545 0.86 CCR5 (0.53) CCR5CCR2CCR7CXCR3
SCHEMBL7216414 0.84 CCR5 (0.54) CCR5
SCHEMBL7216631 0.83 CCR5 (0.51) CCR5CCR2
SCHEMBL7222389 0.81 ACHE (0.54) CCR5
SCHEMBL7221955 0.81 CCR5 (0.47) CCR5
SCHEMBL7216092 0.81 CCR5 (0.51) CCR5CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
US-20030078189-A1 Medicinal compositions for oral use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2003-04-24 US disclosed
EP-1236476-A1 MEDICINAL COMPOSITIONS FOR ORAL USE Takeda Chemical Industries, Ltd. (JP) 2002-09-04 EP disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030078189-A1 Medicinal compositions for oral use CCR5, CXCR3, CCL5 CCR5 1/4885CCR2 23/4885CCR7 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.