SCHEMBL7169161

SCHEMBL7169161

CC(C)(C)OC(=O)N1C[C@H](O)C[C@H]1C(=O)N(CCCN1CCC(Cc2ccccc2)CC1)Cc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.49
CCR5 P51681 1/20 0.45
LMNA P02545 2/20 0.43
KDM4E B2RXH2 2/20 0.43
GAA P10253 1/20 0.43
CCR3 P51677 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KCNH2 Q12809 1/20 0.40
ALDH1A1 P00352 1/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4777983 0.84 OPRM1 (0.48) OPRM1CCR5LMNAKDM4EGAA
Trifluoroacetic Acid SCHEMBL4773894 0.79 CCR5 (0.55) OPRM1CCR5LMNAKDM4EGAA
SCHEMBL6691355 0.79 ALDH1A1 (0.46) LMNAKDM4EHRH3TP53MAPT
SCHEMBL7142421 0.79 ALDH1A1 (0.46) LMNAKDM4EHRH3TP53MAPT
SCHEMBL16836177 0.76 POLB (0.43) TP53MEN1KMT2AALDH1A1JAK2
SCHEMBL16836174 0.76 POLB (0.43) TP53MEN1KMT2AALDH1A1JAK2
SCHEMBL7455496 0.75 OPRM1 (0.58) OPRM1CCR5LMNAKDM4EGAA
SCHEMBL4775520 0.73 GAA (0.57) OPRM1CCR5LMNAKDM4EGAA
SCHEMBL4773843 0.72 OPRM1 (0.49) OPRM1CCR5LMNAKDM4EGAA
Trifluoroacetic Acid SCHEMBL7163436 0.72 OPRM1 (0.49) OPRM1CCR5LMNAKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed