SCHEMBL7175309

SCHEMBL7175309

CCCCCC1=C(CC(=O)OCC)CCC1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
RECQL P46063 1/20 0.38
HIF1A Q16665 1/20 0.38
GAA P10253 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
NR4A1 P22736 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
BRD4 O60885 1/20 0.35
NAAA Q02083 1/20 0.35
DGKA P23743 1/20 0.35
SCD O00767 1/20 0.35
CDC25A P30304 6/20 0.35
CDC25B P30305 6/20 0.35
CDC25C P30307 5/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2142693 0.88 ALDH1A1 (0.38) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL7202715 0.86 TSHR (0.48) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL4237197 0.83 ALDH1A1 (0.46) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL8429054 0.82 ALOX5 (0.44) ALDH1A1TDP1LMNAPPARGMAPT
Lithium Ion SCHEMBL8677043 0.80 GPR84 (0.46) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL7187409 0.78 SCD (0.40) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL4297676 0.77 ALDH1A1 (0.40) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL4441878 0.77 ALDH1A1 (0.39) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL11760628 0.75 SCD (0.45) ALDH1A1TDP1LMNAPOLBRECQL
SCHEMBL11766118 0.75 SCD (0.45) ALDH1A1TDP1LMNAPOLBRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0920354-B1 RUTHENIUM CATALYSTS AND THEIR USE IN THE ASYMMETRIC HYDROGENATION OF WEAKLY COORDINATING SUBSTRATES FIRMENICH & CIE (CH) 2003-12-03 EP disclosed
US-6455460-B1 RU COMPLEX, A BIDENTATE DIPHOSPHINE LIGAND, ACID (HBF4, HPF6, HSBF6, HASF6, HB(3,5-(CF3)2 C6H4); ISOMER OF HEDIONE? OF +(1R)-CIS CONFIGURATION; ASYMMETRIC HYDROGENATION OF HIGHLY HINDERED CARBON-CARBON DOUBLE BONDS FIRMENICH SA (CH) 2002-09-24 US disclosed
US-6214763-B1 HYDROGENATION CATALYST WITH DIPHOSPHINE AND ACID FIRMENICH SA (CH) 2001-04-10 US disclosed
EP-0920354-A1 RUTHENIUM CATALYSTS AND THEIR USE IN THE ASYMMETRIC HYDROGENATION OF WEAKLY COORDINATING SUBSTRATES FIRMENICH SA (CH) 1999-06-09 EP disclosed
WO-1998052687-A1 RUTHENIUM CATALYSTS AND THEIR USE IN THE ASYMMETRIC HYDROGENATION OF WEAKLY COORDINATING SUBSTRATES FIRMENICH S.A. (CH) 1998-11-26 WO disclosed