SCHEMBL7176972

SCHEMBL7176972

CCCCCN(C)CCCCCCOc1ccc(N(C)C(=S)Nc2ccc(Br)cc2C)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPY1R P25929 1/20 0.44
NPY2R P49146 1/20 0.44
LSS P48449 6/20 0.42
PTGES O14684 1/20 0.41
NPC1 O15118 2/20 0.38
THRA P10827 3/20 0.37
THRB P10828 3/20 0.37
PLK1 P53350 2/20 0.37
MMP1 P03956 1/20 0.37
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
ADAM17 P78536 1/20 0.37
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36
NR5A1 Q13285 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3369705 0.88 LSS (0.54) LSS
SCHEMBL7176866 0.79 PTGES (0.52) PTGES
SCHEMBL7207718 0.76 NPY1R (0.41) NPY1RNPY2RLSS
SCHEMBL3367508 0.70 LSS (0.51) LSSPTGES
SCHEMBL7169877 0.69 THRA (0.51) LSSTHRATHRBNR5A1
SCHEMBL7166938 0.69 THRA (0.51) LSSTHRATHRBNR5A1
SCHEMBL3369726 0.69 LSS (0.52) LSSPTGES
SCHEMBL5452892 0.68 NR5A1 (0.54) PTGESNPC1THRATHRBNR5A1
SCHEMBL7165071 0.67 THRA (0.47) LSSTHRATHRB
SCHEMBL16968358 0.67 NR5A1 (0.56) LSSNPC1THRATHRBNR5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303503-A2 ANILINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2002006189-A2 ANILINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-01-24 WO disclosed