SCHEMBL7179028

SCHEMBL7179028

CC=CC(C)Oc1ccc(C=O)c(OC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.61
CYP1A1 P04798 5/20 0.44
CYP1A2 P05177 5/20 0.44
CYP1B1 Q16678 5/20 0.44
MAPT P10636 3/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
ERN1 O75460 1/20 0.42
TRIM24 O15164 1/20 0.41
TYR P14679 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
TNFRSF1A P19438 1/20 0.40
NFE2L2 Q16236 1/20 0.40
MAOB P27338 2/20 0.39
MAPK1 P28482 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3633730 0.83 ALDH1A1 (0.71) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL7184478 0.81 TYR (0.57) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL18478003 0.80 ALDH1A1 (0.67) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL96291 0.77 ALDH1A1 (1.00) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL11774313 0.77 ALDH1A1 (0.61) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL8356166 0.76 ALDH1A1 (0.75) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
Hydrochloric Acid SCHEMBL9456784 0.76 ALDH1A1 (0.96) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL29136568 0.75 ALDH1A1 (0.59) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL5566174 0.75 ALDH1A1 (0.80) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT
SCHEMBL29136540 0.74 ALDH1A1 (0.73) ALDH1A1CYP1A1CYP1A2CYP1B1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-B1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA LICA PHARMACEUTICALS AS (DK) 2001-07-04 EP disclosed
US-5985935-A PARASITICIDES OR BACTERICIDES STATENS SERUMINSTITUT (DK) 1999-11-16 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed