SCHEMBL7181785

SCHEMBL7181785

CC(C)(C)OC(=O)CNCCc1ccc2c(c1)NC(=S)C1(F)CCCC21

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.40
NOS1 P29475 3/20 0.40
NOS2 P35228 3/20 0.40
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
CYP2D6 P10635 3/20 0.31
S1PR1 P21453 1/20 0.31
PKM P14618 1/20 0.30
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30
DPP4 P27487 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
KCNH2 Q12809 1/20 0.30
IGF1R P08069 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6137714 0.91 NOS3 (0.40) NOS3NOS1NOS2KDM4EALDH1A1
SCHEMBL7171051 0.91 NOS3 (0.39) NOS3NOS1NOS2HRH3S1PR1
SCHEMBL6137660 0.82 NOS3 (0.39) NOS3NOS1NOS2HRH3S1PR1
SCHEMBL7145257 0.68 NPC1 (0.50) ALDH1A1HRH3PKMMEN1KMT2A
SCHEMBL7148179 0.67 TAAR1 (0.50) NOS3NOS1KDM4EMEN1KMT2A
SCHEMBL11385307 0.67 MTNR1A (0.56) KDM4EALDH1A1PKM
SCHEMBL6137525 0.67 NOS3 (0.41) NOS3NOS1NOS2
SCHEMBL7135245 0.67 ALDH1A1 (0.48) KDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL7456281 0.66 SPR (0.51) KDM4ECYP2D6KCNH2
SCHEMBL15876078 0.64 SLC7A5 (0.52) CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6579883-B1 Nitrogen monoxide synthases; 4-amino-8-bromo-3a-fluoro-2,3,3a,9b-tetrahydro-1H-cyclopenta (c) quinoline; neurodegenerative, autoimmune, cardiovascular diseases SCHERING AKTIENGESELLSCHAFT (DE) 2003-06-17 US disclosed