SCHEMBL7181983

SCHEMBL7181983

COC(=O)c1ccc2c(c1)c(=O)n(Cc1ccc(F)c(Cl)c1)c(=O)n2C

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARG Q86W56 2/20 0.48
MMP13 P45452 1/20 0.47
SLC22A8 Q8TCC7 1/20 0.47
HDAC1 Q13547 3/20 0.47
TP53 P04637 1/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC8 Q9BY41 1/20 0.45
MAPT P10636 3/20 0.42
P2RX3 P56373 2/20 0.42
MEN1 O00255 1/20 0.42
CASP3 P42574 1/20 0.42
KMT2A Q03164 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
P2RX7 Q99572 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7105312 0.91 PARG (0.48) PARGMMP13SLC22A8HDAC1TP53
SCHEMBL27588029 0.90 PARG (0.52) PARGMMP13SLC22A8HDAC1TP53
SCHEMBL7012164 0.89 MMP13 (0.56) PARGMMP13SLC22A8HDAC1HDAC6
SCHEMBL27588034 0.89 PARG (0.52) PARGMMP13SLC22A8HDAC1TP53
SCHEMBL7018812 0.85 MAPT (0.53) MMP13HDAC1HDAC6HDAC8MAPT
SCHEMBL7660115 0.85 MAPT (0.57) HDAC1TP53MAPTMEN1KMT2A
SCHEMBL7103213 0.84 PARG (0.52) PARGMMP13SLC22A8HDAC1TP53
SCHEMBL7634243 0.84 TP53 (0.57) PARGMMP13SLC22A8HDAC1TP53
SCHEMBL27588009 0.84 PARG (0.54) PARGMMP13SLC22A8HDAC1TP53
SCHEMBL27588021 0.84 PARG (0.54) PARGMMP13SLC22A8HDAC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1537105-A Quinazolines useful as MMP-13 inhibitors ��������ʲ��������ι�˾ 2004-10-13 CN disclosed
EP-1368324-A1 QUINAZOLINES AS MMP-13 INHIBITORS Warner-Lambert Company LLC (US) 2003-12-10 EP disclosed
US-20020193377-A1 Quinazolines as MMP-13 inhibitors ANDRIANJARA CHARLES (FR) 2002-12-19 US disclosed
WO-2002064572-A1 QUINAZOLINES AS MMP-13 INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020193377-A1 Quinazolines as MMP-13 inhibitors MMP13, MMP9, MMP3 PARG 3624/4885MMP13 1/4885SLC22A8 315/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.