Prochlorperazine

Prochlorperazine

SCHEMBL718254

CN1CCN(CCCN2c3ccccc3Sc3ccc(Cl)cc32)CC1.O=C(O)C=CC(=O)O.O=C(O)C=CC(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Prochlorperazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 9/20 0.82
LMNA P02545 8/20 1.00
MAPT P10636 7/20 1.00
MAPK1 P28482 6/20 1.00
SMN1; SMN2 Q16637 5/20 1.00
NPSR1 Q6W5P4 4/20 1.00
MEN1 O00255 4/20 1.00
KMT2A Q03164 4/20 1.00
KDM4E B2RXH2 3/20 1.00
GMNN O75496 3/20 1.00
PMP22 Q01453 3/20 1.00
GAA P10253 1/20 1.00
CYP3A4 P08684 7/20 0.82
ADRA2A P08913 7/20 0.82
ADRA2C P18825 7/20 0.82
SLC6A2 P23975 7/20 0.82
HTR2A P28223 7/20 0.82
SLC6A4 P31645 7/20 0.82
HRH1 P35367 7/20 0.82
DRD3 P35462 7/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prochlorperazine SCHEMBL8911628 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL29686418 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL8914157 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL29634451 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL5494383 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL40755 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL1806022 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL40756 1.00 LMNA (1.00) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Prochlorperazine SCHEMBL28763049 0.95 LMNA (0.91) LMNAMAPTMAPK1SMN1; SMN2NPSR1
Perphenazine SCHEMBL871706 0.92 MAPT (0.85) LMNAMAPTMAPK1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 214 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024028324-A1 MOLECULES FOR THE PREVENTION AND TREATMENT OF NEUROMUSCULAR DISORDERS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2024-02-08 WO claimed
WO-2018039159-A1 MUSCARINIC M2-ANTAGONIST COMBINATION CHASE PHARMACEUTICALS CORPORATION (US) 2018-03-01 WO claimed
WO-2017147104-A1 MUSCARINIC M2-ANTAGONIST COMBINATIONS CHASE PHARMACEUTICALS CORPORATION (US) 2017-08-31 WO claimed
US-20110224141-A1 METHODS AND RELATED COMPOSITIONS FOR THE TREATMENT OF CANCER STC.UNM (US) 2011-09-15 US claimed
WO-2009148623-A2 METHODS AND RELATED COMPOSITIONS FOR THE TREATMENT OF CANCER STC.UNM (US) 2009-12-10 WO claimed
CN-122094715-A Peptide nanosponges for drug delivery 2026-05-26 CN disclosed
US-20250340671-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR REDUCING THE NEUROMODULATORY EFFECT OF COCAINE UNIVERSITY OF CINCINNATI (US) 2025-11-06 US disclosed
US-20240197728-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR TREATING REFRACTORY EPILEPSY INST NAT SANTE RECH MED (FR) 2024-06-20 US disclosed
EP-4322952-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR TREATING REFRACTORY EPILEPSY Inserm (Institut National de la Santé et de la Recherche Scientifique) (FR) 2024-02-21 EP disclosed
WO-2024028324-A1 MOLECULES FOR THE PREVENTION AND TREATMENT OF NEUROMUSCULAR DISORDERS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2024-02-08 WO disclosed
WO-2023235500-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR REDUCING THE NEUROMODULATORY EFFECT OF COCAINE UNIVERSITY OF CINCINNATI (US) 2023-12-07 WO disclosed
US-11759445-B2 Use of Rivastigmine in preparation of anti-radiation medicament SOOCHOW UNIVERSITY (CN) 2023-09-19 US disclosed
US-5654281-A Inhibiting the development of tolerance to and/or dependence on an addictive substance VIRGINIA COMMONWEALTH UNIVERSITY (US) 1997-08-05 US disclosed
EP-0778770-A1 COMPOSITION ALLEVIATING PAIN, CONTAINING A NON-NARCOTIC ANALGESIC AND AN ANALGESIA ENHANCER VIRGINIA COMMONWEALTH UNIVERSITY (US) 1997-06-18 EP disclosed
US-5556838-A BLOCKING N-METHYLASPARTATE RECEPTORS TO PREVENT ADDICTION VIRGINIA COMMONWEALTH UNIVERSITY (US) 1996-09-17 US disclosed
US-5502058-A Method for the treatment of pain VIRGINIA COMMONWEALTH UNIVERSITY (US) 1996-03-26 US disclosed
WO-1996007412-A1 COMPOSITION ALLEVIATING PAIN, CONTAINING A NON-NARCOTIC ANALGESIC AND AN ANALGESIA ENHANCER VIRGINIA COMMONWEALTH UNIVERSITY (US) 1996-03-14 WO disclosed
EP-0615749-A2 Use of NMDA antagonists for the treatment of pain VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-09-21 EP disclosed
EP-0608893-A1 Inhibiting the development of tolerance to and/or dependence on an additive substance VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-08-03 EP disclosed
US-5321012-A Inhibiting the development of tolerance to and/or dependence on a narcotic addictive substance VIRGINIA COMMONWEALTH UNIVERSITY MEDICAL COLLEGE (US) 1994-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240197728-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR TREATING REFRACTORY EPILEPSY SLC6A13, SLC6A1, CLCN2 DRD2 1213/4885LMNA 3265/4885MAPT 1619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.