Malonic Acid

Malonic Acid

SCHEMBL718362

NC(CO)CO.O=C(O)CC(=O)O

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.53
SRR Q9GZT4 1/20 0.53
ENPEP Q07075 7/20 0.37
ANPEP P15144 3/20 0.37
SLC1A1 P43005 2/20 0.37
USP2 O75604 1/20 0.36
SLCO1B1 Q9Y6L6 1/20 0.36
OR51E2 Q9H255 2/20 0.35
GLRA1 P23415 1/20 0.35
SLC6A9 P48067 1/20 0.35
GABRP O00591 2/20 0.35
GABRD O14764 2/20 0.35
GABRA1 P14867 2/20 0.35
GABRB1 P18505 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA5 P31644 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRB2 P47870 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Malonic Acid SCHEMBL25382800 0.92 LDHA (0.45) LDHASRRENPEPANPEPSLC1A1
Glycolic Acid SCHEMBL22346352 0.85 ENPEP (0.39) ENPEPANPEPSLC1A1USP2SLCO1B1
Succinic Acid SCHEMBL22346000 0.82 LMNA (0.53) ENPEPANPEPSLC1A1OR51E2GABRP
Oxalic Acid SCHEMBL7088814 0.81 SLC1A1 (0.40) LDHAENPEPANPEPSLC1A1USP2
Carbamic Acid SCHEMBL27083006 0.81 ACHE (0.47) LDHAENPEPANPEPSLC1A1USP2
Acetic Acid SCHEMBL7045506 0.79 FFAR3 (0.44) ENPEPANPEPSLC1A1USP2SLCO1B1
SCHEMBL2354479 0.77 LMNA (0.36) SLC1A1
SCHEMBL74076 0.77
SCHEMBL3895147 0.77
SCHEMBL288980 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240189263-A1 DERIVATIZED C60 MOLECULES AND METHODS AND MATERIALS FOR USING DERIVATIZED C60 MOLECULES TO REDUCE RADIATION INJURY MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2024-06-13 US claimed
WO-2023167700-A9 DERIVATIZED C60 MOLECULES AND METHODS AND MATERIALS FOR USING DERIVATIZED C60 MOLECULES TO REDUCE RADIATION INJURY MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2023-10-19 WO claimed
WO-2023167700-A2 DERIVATIZED C60 MOLECULES AND METHODS AND MATERIALS FOR USING DERIVATIZED C60 MOLECULES TO REDUCE RADIATION INJURY MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2023-09-07 WO claimed
US-20090214101-A1 Targeted Nanostructures for Cellular Imaging WILLIAM MARSH RICE UNIVERSITY 2009-08-27 US claimed
US-20080175892-A1 Nanostructure-Drug Conjugates WILLIAM MARSH RICE UNIVERSITY 2008-07-24 US claimed
WO-2007143558-A1 TARGETED NANOSTRUCTURES FOR CELLULAR IMAGING WILLIAM MARSH RICE UNIVERSITY (US) 2007-12-13 WO claimed
US-20240189263-A1 DERIVATIZED C60 MOLECULES AND METHODS AND MATERIALS FOR USING DERIVATIZED C60 MOLECULES TO REDUCE RADIATION INJURY MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2024-06-13 US disclosed
WO-2023167700-A9 DERIVATIZED C60 MOLECULES AND METHODS AND MATERIALS FOR USING DERIVATIZED C60 MOLECULES TO REDUCE RADIATION INJURY MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2023-10-19 WO disclosed
WO-2023167700-A2 DERIVATIZED C60 MOLECULES AND METHODS AND MATERIALS FOR USING DERIVATIZED C60 MOLECULES TO REDUCE RADIATION INJURY MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2023-09-07 WO disclosed
US-8986942-B2 Carbon nanotube based imaging agents WILLIAM MARSH RICE UNIVERSITY (US) 2015-03-24 US disclosed
US-20130130295-A1 CARBON NANOTUBE BASED IMAGING AGENTS WILLIAM MARSH RICE UNIVERSITY 2013-05-23 US disclosed
US-20120141543-A1 Carbon Nanotube Based Nanocomposites NATIONAL SCIENCE FOUNDATION 2012-06-07 US disclosed
US-20120052004-A1 CARBON NANOTUBE BASED MAGNETIC RESONANCE IMAGE CONTRAST AGENTS WILLIAM MARSH RICE UNIVERSITY 2012-03-01 US disclosed
WO-2011019882-A1 NANOSTRUCTURE-BETA-BLOCKER CONJUGATES WILLIAM MARSH RICE UNIVERSITY (US) 2011-02-17 WO disclosed
WO-2010017546-A1 CARBON NANOTUBE BASED MAGNETIC RESONANCE IMAGING CONTRAST AGENTS WILLIAM MARSH RICE UNIVERSITY (US) 2010-02-11 WO disclosed
US-20090214101-A1 Targeted Nanostructures for Cellular Imaging WILLIAM MARSH RICE UNIVERSITY 2009-08-27 US disclosed
US-20090136987-A1 Carbon Nanotube Based Imaging Agents WILSON LON J 2009-05-28 US disclosed
US-20080175892-A1 Nanostructure-Drug Conjugates WILLIAM MARSH RICE UNIVERSITY 2008-07-24 US disclosed
WO-2007143558-A1 TARGETED NANOSTRUCTURES FOR CELLULAR IMAGING WILLIAM MARSH RICE UNIVERSITY (US) 2007-12-13 WO disclosed
WO-2007137256-A2 CARBON NANOTUBE BASED IMAGING AGENTS WILLIAM MARSH RICE UNIVERSITY (US) 2007-11-29 WO disclosed