SCHEMBL7185508

SCHEMBL7185508

COC(=O)C(=O)C(C=O)c1cc2ccccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP6V1B1 P15313 1/20 0.48
ALOX5 P09917 1/20 0.46
KDM4E B2RXH2 3/20 0.43
LMNA P02545 2/20 0.43
TP53 P04637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
DRD2 P14416 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
FLT3 P36888 4/20 0.41
CYP2A6 P11509 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PDGFRB P09619 2/20 0.40
PDGFRA P16234 2/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
HPGD P15428 2/20 0.40
MAPT P10636 1/20 0.40
DAO P14920 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7193003 0.84 KDM4E (0.46) ALOX5KDM4ELMNATP53L3MBTL1
SCHEMBL2661862 0.81 KDM4E (0.49) ALOX5KDM4ELMNATP53L3MBTL1
SCHEMBL12827519 0.72 ALOX5 (0.51) ALOX5KDM4ELMNATP53L3MBTL1
SCHEMBL29933860 0.71 DRD2 (0.52) ATP6V1B1ALOX5KDM4ELMNATP53
SCHEMBL9337151 0.71 KDM4E (0.47) ALOX5KDM4ELMNATP53L3MBTL1
SCHEMBL5957825 0.70 FLT3 (0.61) ATP6V1B1KDM4ELMNATP53L3MBTL1
SCHEMBL28692760 0.69 CYP2A6 (0.50) ALOX5KDM4ELMNATP53L3MBTL1
SCHEMBL2350318 0.69 ALOX5 (0.55) ALOX5KDM4ELMNATP53L3MBTL1
SCHEMBL3329679 0.69 FLT3 (0.59) ATP6V1B1KDM4ELMNATP53L3MBTL1
SCHEMBL7185518 0.69 IDO1 (0.56) KDM4ELMNATP53L3MBTL1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1083897-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-01-02 EP claimed
EP-1083897-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-21 EP claimed
WO-1999062513-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO claimed
EP-1083897-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2003-01-02 EP disclosed
EP-1083897-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2001-03-21 EP disclosed
WO-1999062513-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 1999-12-09 WO disclosed