SCHEMBL7187230

SCHEMBL7187230

Cc1ncn(-c2nc(C(N)=O)c(O)c(=O)n2C)n1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.34
FEN1 P39748 1/20 0.34
ERCC4 Q92889 1/20 0.34
MEN1 O00255 1/20 0.32
PABPC1 P11940 1/20 0.32
KMT2A Q03164 1/20 0.32
TRPA1 O75762 2/20 0.32
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
LMNA P02545 2/20 0.30
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6095015 0.83 LMNA (0.39) ADORA2AADORA1LMNAALDH1A1MAPT
SCHEMBL6094959 0.75 KCNE1 (0.51) ERCC1FEN1ERCC4MEN1KMT2A
SCHEMBL6092877 0.73 CNR1 (0.46)
SCHEMBL6093853 0.72 MMP13 (0.47) MEN1KMT2A
SCHEMBL6883899 0.66 MEN1 (0.44) MEN1PABPC1KMT2AADORA2AADORA1
SCHEMBL18832230 0.64 ERCC1 (0.36) ERCC1FEN1ERCC4LMNAALDH1A1
SCHEMBL27803655 0.62 ALDH1A1 (0.43) LMNAALDH1A1MAPT
SCHEMBL30621294 0.60 KDM4E (0.61) MEN1KMT2AALDH1A1MAPT
SCHEMBL17825684 0.60 NPC1 (0.44) ADORA2AADORA1LMNAALDH1A1MAPT
SCHEMBL5766494 0.60 KMT2A (0.40) MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004062613-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-07-29 WO disclosed