SCHEMBL7189809

SCHEMBL7189809

CCOP(=O)(OCC)c1cccc(CCCBr)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
LTA4H P09960 1/20 0.37
EPHX2 P34913 1/20 0.37
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
POLB P06746 1/20 0.36
ACHE P22303 1/20 0.36
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4411677 0.88 NPSR1 (0.47) NPSR1MEN1KMT2ALTA4HEPHX2
SCHEMBL12229723 0.84 NPSR1 (0.45) NPSR1MEN1KMT2ALTA4HEPHX2
SCHEMBL8116136 0.82 LTA4H (0.42) NPSR1MEN1KMT2ACYP4F2CYP4A11
SCHEMBL12229683 0.81 POLB (0.53) NPSR1MEN1KMT2ALTA4HEPHX2
SCHEMBL12229697 0.78 NPSR1 (0.45) NPSR1MEN1KMT2ALTA4HEPHX2
SCHEMBL7525626 0.78 CYP4F2 (0.44) NPSR1MEN1KMT2ACYP4F2CYP4A11
SCHEMBL9849286 0.75 LMNA (0.42) NPSR1MEN1KMT2ACYP4F2CYP4A11
SCHEMBL9849259 0.75 NPC1 (0.45) MEN1KMT2ALTA4HEPHX2CA12
SCHEMBL14809313 0.75 MEN1 (0.48) NPSR1MEN1KMT2ALTA4HEPHX2
SCHEMBL12229745 0.75 MEN1 (0.48) NPSR1MEN1KMT2ALTA4HEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268494-A1 SULFUR SUBSTITUTED ARYLDIFLUOROMETHYLPHOSPHONIC ACIDS AS PTP-1B INHIBITORS Merck Frosst Canada & Co. (CA) 2003-01-02 EP disclosed
WO-2001070753-A1 SULFUR SUBSTITUTED ARYLDIFLUOROMETHYLPHOSPHONIC ACIDS AS PTP-1B INHIBITORS MERCK FROSST CANADA & CO. (CA) 2001-09-27 WO disclosed