Benzenesulfonamide

Benzenesulfonamide

SCHEMBL7192191

COc1ccc(-c2cc(C(F)(F)F)nn2NS(=O)(=O)c2ccccc2)cc1F.NS(=O)(=O)c1ccccc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.53
PTGS1 P23219 14/20 0.52
ABCB11 O95342 1/20 0.48
ALDH1A1 P00352 1/20 0.48
PDPK1 O15530 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640455 0.95 PTGS2 (0.45) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8692192 0.88 PTGS2 (0.42) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8689604 0.87 PTGS2 (0.41) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8637024 0.87 PTGS2 (0.54) PTGS2PTGS1
Benzenesulfonamide SCHEMBL8525050 0.86 PTGS2 (0.61) PTGS2PTGS1PDPK1
Benzenesulfonamide SCHEMBL7046453 0.86 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8639246 0.85 PTGS2 (0.56) PTGS2PTGS1ALDH1A1
SCHEMBL7775609 0.85 PTGS2 (0.55) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8636828 0.85 PDPK1 (0.61) PTGS2PTGS1ABCB11PDPK1
SCHEMBL8689324 0.84 PTGS2 (0.45) PTGS2PTGS1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001505564-A 2001-04-24 JP claimed
EP-0941080-A2 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS AS ANTI-ANGIOGENIC AGENTS G.D. SEARLE & CO. (US) 1999-09-15 EP claimed
WO-1998022101-A2 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS AS ANTI-ANGIOGENIC AGENTS G.D. SEARLE & CO. (US) 1998-05-28 WO claimed
EP-1365753-A2 UROGUANYLIN AND CYCLOOXYGENASE-2 INHIBITOR COMBINATIONS FOR INHIBITION OF INTESTINAL CANCER Pharmacia Corporation (US) 2003-12-03 EP disclosed
WO-2002062369-A2 UROGUANYLIN AND CYCLOOXYGENASE-2 INHIBITOR COMBINATIONS FOR INHIBITION OF INTESTINAL CANCER PHARMACIA CORPORATION (US) 2002-08-15 WO disclosed
EP-0979077-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. Searle & Co. (US) 2000-02-16 EP disclosed
WO-1998047509-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE PREVENTION OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1998-10-29 WO disclosed