SCHEMBL7775609

SCHEMBL7775609

COc1ccc(-c2cc(C(F)(F)F)nn2NS(=O)(=O)c2ccccc2)cc1F.COc1ccc(-c2cc(C(F)F)nn2-c2ccccc2S(N)(=O)=O)cc1F

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.55
PTGS1 P23219 10/20 0.55
ABCB11 O95342 1/20 0.55
ALDH1A1 P00352 1/20 0.55
F10 P00742 2/20 0.38
F2 P00734 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8385316 0.86 PTGS2 (0.69) PTGS2PTGS1ABCB11ALDH1A1
Benzenesulfonamide SCHEMBL7192191 0.85 PTGS2 (0.53) PTGS2PTGS1ABCB11ALDH1A1
Benzenesulfonamide SCHEMBL7046453 0.84 PTGS2 (0.65) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7920280 0.84 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8640455 0.84 PTGS2 (0.45) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL7932075 0.83 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8688532 0.79 PTGS2 (0.57) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8692194 0.78 PTGS2 (0.50) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8691591 0.78 PTGS2 (0.57) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL8692192 0.78 PTGS2 (0.42) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2001503395-A 2001-03-13 JP claimed
EP-0932402-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA G.D. SEARLE & CO. (US) 1999-08-04 EP claimed
WO-1998016227-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA G.D. SEARLE & CO. (US) 1998-04-23 WO claimed
EP-0932402-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA G.D. SEARLE & CO. (US) 1999-08-04 EP disclosed
WO-1998016227-A9 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA 1998-07-30 WO disclosed
WO-1998016227-A1 METHOD OF USING CYCLOOXYGENASE-2 INHIBITORS IN THE TREATMENT AND PREVENTION OF NEOPLASIA G.D. SEARLE & CO. (US) 1998-04-23 WO disclosed