SCHEMBL7192547

SCHEMBL7192547

O=c1oc2c[c]ccc2cc1-c1ccc2[nH]cnc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 3/20 0.36
RAB9A P51151 6/20 0.35
ALDH1A1 P00352 6/20 0.35
KDM4E B2RXH2 5/20 0.35
MAOB P27338 2/20 0.35
NPC1 O15118 4/20 0.35
HPGD P15428 4/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
GAPDH P04406 2/20 0.35
GAA P10253 2/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
ESR1 P03372 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MIF P14174 6/20 0.35
TP53 P04637 2/20 0.34
MAPT P10636 3/20 0.34
MEN1 O00255 2/20 0.33
GLA P06280 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3396561 0.73 RAB9A (0.66) ESR2RAB9AALDH1A1KDM4EMAOB
SCHEMBL16720439 0.72 QPCT (0.50) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL3400256 0.71 GAPDH (0.55) ESR2RAB9AALDH1A1KDM4EMAOB
SCHEMBL3398092 0.70 GPR35 (0.48) ESR2RAB9AALDH1A1KDM4EMAOB
SCHEMBL27601236 0.69 QPCT (0.41) RAB9AALDH1A1KDM4ENPC1HPGD
SCHEMBL6928197 0.69 RAB9A (0.73) RAB9AALDH1A1KDM4ENPC1HPGD
SCHEMBL5757411 0.68 MEN1 (0.40) RAB9AALDH1A1KDM4ENPC1HPGD
SCHEMBL8671614 0.68 QPCT (0.38) RAB9AALDH1A1KDM4ENPC1HPGD
SCHEMBL5756878 0.67 QPCT (0.40) RAB9AALDH1A1KDM4ENPC1HPGD
SCHEMBL6931520 0.67 MAPT (0.72) RAB9AALDH1A1KDM4EMAOBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6566355-B1 Useful in combination with beta -lactam antibiotics in the control of beta -lactamase forming pathogens HOFFMANN-LA ROCHE INC. 2003-05-20 US disclosed
US-5510343-A BETA-LACTAMASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-04-23 US disclosed