SCHEMBL7197345

SCHEMBL7197345

FC(F)(F)Oc1c(Cc2ccccc2)nc2n1CCNC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
TAAR1 Q96RJ0 2/20 0.36
HTR6 P50406 1/20 0.36
CYP2D6 P10635 3/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
KCNH2 Q12809 2/20 0.35
HTR2C P28335 7/20 0.34
HTR2A P28223 5/20 0.34
HTR2B P41595 5/20 0.34
LTA4H P09960 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
CETP P11597 1/20 0.33
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
ADRA2A P08913 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7197337 0.83 LIPG (0.39) MCHR1LIPGTAAR1HTR6CYP2D6
SCHEMBL10153396 0.67 TAAR1 (0.48) MCHR1TAAR1HTR6SLC6A2SLC6A4
SCHEMBL10095064 0.65 P2RX7 (0.45) LIPGHTR2CHTR2ACYP1A2TSHR
SCHEMBL5880518 0.62 NR1H4 (0.44)
SCHEMBL29539173 0.61 HTR2A (0.50) MCHR1HTR2CHTR2ATSHR
SCHEMBL839815 0.61 HTR2A (0.50) MCHR1HTR2CHTR2ATSHR
Hydrochloric Acid SCHEMBL20139551 0.60 HTR2A (0.49) MCHR1HTR2CHTR2ATSHR
SCHEMBL28783649 0.60 ADRB2 (0.39) LIPGHTR6HTR2CHTR2AHTR2B
SCHEMBL10095057 0.60 PDCD1 (0.41) MCHR1HTR6CYP2D6HTR2CHTR2A
SCHEMBL24176694 0.59 SLC6A2 (0.43) SLC6A2SLC6A4CYP1A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294700-A2 BENZHYDRYL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-03-26 EP disclosed
WO-2002000631-A2 BENZHYDRYL DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-01-03 WO disclosed