SCHEMBL7200630

SCHEMBL7200630

COc1ccccc1C(=O)C(O)=Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.53
POLB P06746 2/20 0.53
ABCG2 Q9UNQ0 1/20 0.51
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
CA9 Q16790 1/20 0.51
RAB9A P51151 1/20 0.47
CTSD P07339 1/20 0.47
HTT P42858 1/20 0.47
AKR1C3 P42330 1/20 0.46
HPGD P15428 3/20 0.45
TP53 P04637 1/20 0.45
GLA P06280 1/20 0.45
STAT3 P40763 1/20 0.45
GPR52 Q9Y2T5 1/20 0.44
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
PLIN1 O60240 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10741205 0.91 ABCG2 (0.50) NPC1POLBABCG2CA12CA1
SCHEMBL4535104 0.84 NPC1 (0.54) NPC1POLBABCG2CA12CA1
SCHEMBL6576793 0.80 AKR1C2 (0.56) NPC1POLBABCG2CA12CA1
SCHEMBL870484 0.80 CTSD (0.62) NPC1ABCG2CA12CA1CA2
SCHEMBL29242266 0.79 AR (0.48) NPC1POLBABCG2CA12CA1
SCHEMBL4621633 0.78 STAT3 (0.58) NPC1ABCG2CA12CA1CA2
SCHEMBL29875455 0.78 STAT3 (0.58) NPC1ABCG2CA12CA1CA2
SCHEMBL675699 0.77 KDM4E (0.50) NPC1POLBRAB9AAKR1C3HPGD
SCHEMBL11774603 0.77 ALDH1A1 (0.56) POLBCA12CA1CA2CA9
SCHEMBL1073512 0.77 MAPT (0.55) NPC1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6603046-B1 The invention is drawn to novel bis-aromatic a, beta -unsaturated ketones. The compounds are useful in the treatment and prophylaxis of diseases caused by parasites or bacteria. LICA PHARMACEUTICALS A/S (DK) 2003-08-05 US disclosed
EP-0634927-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1995-01-25 EP disclosed
WO-1993017671-A1 TREATMENT AND PROPHYLAXIS OF DISEASES CAUSED BY PARASITES, OR BACTERIA STATENS SERUMINSTITUT (DK) 1993-09-16 WO disclosed