Propiomazine

Propiomazine

SCHEMBL720224

CCC(=O)c1ccc2c(c1)N(CC(C)N(C)C)c1ccccc1S2.[Cl-].[H+]

nearest known ligand 0.96

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Propiomazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 2/20 0.96
CHRM2 P08172 6/20 0.96
HTR1A P08908 6/20 0.96
CHRM1 P11229 6/20 0.96
ADRA1A P35348 6/20 0.96
OPRM1 P35372 6/20 0.96
DRD3 P35462 6/20 0.96
KCNH2 Q12809 6/20 0.96
DRD2 P14416 3/20 0.96
ADRA2B P18089 2/20 0.96
ADRA2C P18825 2/20 0.96
CHRM3 P20309 2/20 0.96
HTR2A P28223 2/20 0.96
HTR2C P28335 2/20 0.96
OPRK1 P41145 2/20 0.96
HTR2B P41595 2/20 0.96
CYP2D6 P10635 7/20 0.64
CYP1A2 P05177 5/20 0.64
HSD17B10 Q99714 4/20 0.64
MTOR P42345 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Propiomazine SCHEMBL29609596 0.98 CHRM2 (1.00) CHRM2HTR1ACHRM1ADRA1AOPRM1
Propiomazine SCHEMBL29370554 0.98 CHRM2 (1.00) CHRM2HTR1ACHRM1ADRA1AOPRM1
(R)-Propiomazine SCHEMBL6910697 0.98 CHRM2 (1.00) CHRM2HTR1ACHRM1ADRA1AOPRM1
Propiomazine SCHEMBL93770 0.98 CHRM2 (1.00) CHRM2HTR1ACHRM1ADRA1AOPRM1
Propiomazine SCHEMBL30903904 0.97 CHRM2 (0.98) CHRM2HTR1ACHRM1ADRA1AOPRM1
Propiomazine SCHEMBL141677 0.97 CHRM2 (0.98) CHRM2HTR1ACHRM1ADRA1AOPRM1
Propiomazine SCHEMBL6372719 0.97 CHRM2 (0.98) CHRM2HTR1ACHRM1ADRA1AOPRM1
Propiomazine SCHEMBL3863991 0.92 CHRM2 (0.88) CHRM2HTR1ACHRM1ADRA1AOPRM1
SCHEMBL10368273 0.86 CHRM2 (0.79) CHRM2HTR1ACHRM1ADRA1AOPRM1
Aceprometazine SCHEMBL142393 0.86 HTR1A (0.79) CHRM2HTR1ACHRM1ADRA1AOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4483487-A1 MLINC Rheinisch-Westfälische Technische Hochschule (RWTH) Aachen (DE) 2025-01-01 EP disclosed
WO-2023161010-A1 MLINC RHEINISCH-WESTFÄLISCHE TECHNISCHE HOCHSCHULE (RWTH) AACHEN (DE) 2023-08-31 WO disclosed
US-10722562-B2 Combinatorial analysis and repair IMMUDEX APS (DK) 2020-07-28 US disclosed
US-20160361356-A1 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR ENHANCING SURVIVABILITY OF CELLS, TISSUES, ORGANS, AND ORGANISMS FRED HUTCHINSON CANCER RESEARCH CENTER 2016-12-15 US disclosed
EP-2949212-A1 USE OF OXYGEN ANTAGONISTS FOR EX VIVO PRESERVATION OF TISSUES OR ORGANS Fred Hutchinson Cancer Research Center (US) 2015-12-02 EP disclosed
US-20150164064-A1 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN CELLS, TISSUES, ORGANS, AND ORGANISMS FRED HUTCHINSON CANCER RESEARCH CENTER 2015-06-18 US disclosed
US-8822535-B2 Methods, compositions and articles of manufacture for enhancing survivability of cells, tissues, organs, and organisms FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2014-09-02 US disclosed
CN-1901795-B Methods, compositions and devices for inducing stasis in cells, tissues, organs, and organisms HUTCHINSON FRED CANCER RES 2014-03-26 CN disclosed
EP-1879599-B1 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR ENHANCING SURVIVABILITY OF CELLS, TISSUES, ORGANS, AND ORGANISMS HUTCHINSON FRED CANCER RES (US) 2013-10-16 EP disclosed
US-20120282353-A1 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR HIF MODULATING COMPOUNDS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2012-11-08 US disclosed
EP-1689228-A2 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN CELLS Fred Hutchinson Cancer Research Center (US) 2006-08-16 EP disclosed
EP-1684580-A2 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN TISSUES AND ORGANS Fred Hutchinson Cancer Research Center (US) 2006-08-02 EP disclosed
EP-1684579-A1 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN CELLS, TISSUES, ORGANS, AND ORGANISMS Fred Hutchinson Cancer Research Center (US) 2006-08-02 EP disclosed
US-20050170019-A1 Methods, compositions and devices for inducing stasis in cells FRED HUTCHINSON CANCER RESEARCH CENTER 2005-08-04 US disclosed
US-20050147692-A1 Methods, compositions and devices for inducing stasis in tissues and organs FRED HUTCHINSON CANCER RESEARCH CENTER 2005-07-07 US disclosed
US-20050136125-A1 Methods, compositions and devices for inducing stasis in cells, tissues, organs, and organisms NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-06-23 US disclosed
WO-2005041655-A1 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN CELLS, TISSUES, ORGANS, AND ORGANISMS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2005-05-12 WO disclosed
WO-2005041656-A2 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN TISSUES AND ORGANS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2005-05-12 WO disclosed
WO-2005039291-A2 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN CELLS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2005-05-06 WO disclosed
US-6650679-B1 Preionization arrangement for gas laser LAMBDA PHYSIK AG (DE) 2003-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160361356-A1 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR ENHANCING SURVIVABILITY OF CELLS, TISSUES, ORGANS, AND ORGANISMS BCL2, BAX, HSF1 HRH1 2493/4885CHRM2 3210/4885HTR1A 2012/4885
US-20050147692-A1 Methods, compositions and devices for inducing stasis in tissues and organs HIF1A, HIF1AN, PYGL HRH1 2287/4885CHRM2 3064/4885HTR1A 4061/4885
US-20050136125-A1 Methods, compositions and devices for inducing stasis in cells, tissues, organs, and organisms HSF1, HSP90AB1, HSP90AA1 HRH1 1709/4885CHRM2 3821/4885HTR1A 3278/4885
US-20120282353-A1 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR HIF MODULATING COMPOUNDS HIF1A, HIF1AN, EGLN3 HRH1 2221/4885CHRM2 4789/4885HTR1A 3939/4885
US-20050170019-A1 Methods, compositions and devices for inducing stasis in cells PLAT, TBXA2R, THPO HRH1 3316/4885CHRM2 3976/4885HTR1A 2983/4885
US-20150164064-A1 METHODS, COMPOSITIONS AND DEVICES FOR INDUCING STASIS IN CELLS, TISSUES, ORGANS, AND ORGANISMS HSF1, HSP90AB1, HSP90AA1 HRH1 1709/4885CHRM2 3821/4885HTR1A 3278/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.