5-Chloroindole-2-Carboxylic Acid

5-Chloroindole-2-Carboxylic Acid

SCHEMBL720582

O=C(O)c1cc2cc(Cl)ccc2[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F7 P08709 1/20 1.00
F3 P13726 1/20 1.00
MEN1 O00255 3/20 0.69
KMT2A Q03164 3/20 0.69
NPC1 O15118 1/20 0.69
RAB9A P51151 1/20 0.69
SMAD3 P84022 1/20 0.66
KDM4E B2RXH2 3/20 0.64
HPGD P15428 3/20 0.64
HSD17B10 Q99714 2/20 0.64
LMNA P02545 2/20 0.64
PIN1 Q13526 1/20 0.64
PDPK1 O15530 1/20 0.64
ALDH1A1 P00352 1/20 0.64
TSHR P16473 1/20 0.64
NFKB1 P19838 1/20 0.64
APEX1 P27695 1/20 0.64
CYP2C19 P33261 1/20 0.64
TDP1 Q9NUW8 1/20 0.64
NHERF1 O14745 3/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
5-Chloroindole-2-Carboxylic Acid SCHEMBL6921825 0.98 F7 (0.96) F7F3MEN1KMT2ANPC1
5-Chloroindole-2-Carboxylic Acid SCHEMBL27410586 0.91 F7 (0.82) F7F3MEN1KMT2ANPC1
5-Chloroindole-2-Carboxylic Acid SCHEMBL6162690 0.88 F7 (0.77) F7F3MEN1KMT2ANPC1
SCHEMBL3499567 0.86 F7 (0.76) F7F3MEN1KMT2ANPC1
SCHEMBL30310328 0.85 F7 (0.74) F7F3MEN1KMT2AKDM4E
SCHEMBL671001 0.85 F7 (0.74) F7F3MEN1KMT2AKDM4E
SCHEMBL2694131 0.85 F7 (0.74) F7F3MEN1KMT2ANPC1
SCHEMBL6343336 0.84 F7 (0.72) F7F3MEN1KMT2ANPC1
SCHEMBL2729831 0.84 F7 (0.72) F7F3MEN1KMT2ANPC1
SCHEMBL764543 0.84 F7 (0.72) F7F3MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1365 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118994223-A Aluminum oxide nanotube crystalline material and preparation method and application thereof 中国科学院福建物质结构研究所 2024-11-22 CN claimed
CN-108350034-B Antimicrobial polymyxin derived compounds 莫纳什大学 2022-03-11 CN claimed
US-20220048979-A1 TREATMENT OF STAPHYLOCOCCAL DISORDERS THE UNITED STATES GOVERNMENT AS REPRESENTED BY THE DEPARTMENT OF VETERAN AFFAIRS 2022-02-17 US claimed
EP-1469833-B1 METHOD FOR MAKING HOMOGENEOUS SPRAY-DRIED SOLID AMORPHOUS DRUG DISPERSIONS UTILIZING MODIFIED SPRAY-DRYING APPARATUS BEND RES INC (US) 2021-05-19 EP claimed
CN-109212052-B Gas chromatography-mass spectrometry combined method for measuring five trace indole carboxylic acid compounds in water source water 丁立平 2021-05-11 CN claimed
CN-109212052-A The gas chromatography-mass spectrometry of five kinds of trace indol-carbocylic acids compounds in a kind of measurement source water 丁立平 2019-01-15 CN claimed
EP-2948454-B1 TRIAZINE COMPOUNDS AND A PROCESS FOR PREPARATION THEREOF COUNCIL OF SCIENT & IND RES AN INDIAN REGISTERED BODY INCORPORATED UNDER THE REGISTRATION OF SOCIETI (IN) 2017-05-31 EP claimed
US-20160368928-A1 MELAMPOMAGNOLIDE B DERIVATIVES BIOVENTURES, LLC 2016-12-22 US claimed
CN-103819486-B Photoaffinity probe molecule, its preparation method and the medical usage of labelling serum glycogen phosphorylase concentration level 承德医学院 2016-08-17 CN claimed
US-20150203508-A1 MELAMPOMAGNOLIDE B DERIVATIVES BIOVENTURES, LLC 2015-07-23 US claimed
US-5952322-A AMIDE-SUBSTITUTED BENZIMIDAZOLE, INDOLE DERIVATIVES PFIZER INC. (US) 1999-09-14 US claimed
WO-1999043663-A1 N-[(SUBSTITUTED FIVE-MEMBERED DI- OR TRIAZA DIUNSATURATED RING)CARBONYL] GUANIDINE DERIVATIVES FOR THE TREATMENT OF ISCHEMIA PFIZER PRODUCTS INC. (US) 1999-09-02 WO claimed
WO-1999026659-A1 COMBINATION OF AN ALDOSE REDUCTASE INHIBITOR AND A GLYCOGEN PHOSPHORYLASE INHIBITOR PFIZER PRODUCTS INC. (US) 1999-06-03 WO claimed
EP-0846464-A2 Use of glycogen phosphorylase inhibitor for reducing non-cardiac tissue damage resulting from ischemia PFIZER INC. (US) 1998-06-10 EP claimed
EP-0832065-A1 SUBSTITUTED N-(INDOLE-2-CARBONYL)-GLYCINAMIDES AND DERIVATIVES AS GLYCOGEN PHOSPHORYLASE INHIBITORS PFIZER INC. (US) 1998-04-01 EP claimed
EP-0832066-A1 SUBSTITUTED N-(INDOLE-2-CARBONYL-) AMIDES AND DERIVATIVES AS GLYCOGEN PHOSPHORYLASE INHIBITORS PFIZER INC. (US) 1998-04-01 EP claimed
CN-1140709-A Substituted N- (indole-2-carbonyl) -beta-alaninamides and derivatives as antidiabetics PFIZER (US) 1997-01-22 CN claimed
WO-1996039385-A1 SUBSTITUTED N-(INDOLE-2-CARBONYL-) AMIDES AND DERIVATIVES AS GLYCOGEN PHOSPHORYLASE INHIBITORS PFIZER INC. (US) 1996-12-12 WO claimed
WO-1996039384-A1 SUBSTITUTED N-(INDOLE-2-CARBONYL)-GLYCINAMIDES AND DERIVATIVES AS GLYCOGEN PHOSPHORYLASE INHIBITORS PFIZER, INC. (US) 1996-12-12 WO claimed
US-4123534-A VIGILANCE INCREASING AGENTS Wulfing, Johann W. (DE) 1978-10-31 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150203508-A1 MELAMPOMAGNOLIDE B DERIVATIVES CMBL, MGMT, MMAB F7 3285/4885F3 4734/4885MEN1 220/4885
US-20160368928-A1 MELAMPOMAGNOLIDE B DERIVATIVES CMBL, MGMT, MMAB F7 3285/4885F3 4734/4885MEN1 220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.