SCHEMBL7207972

SCHEMBL7207972

COc1ccc(S(=O)(=O)CCCSNC(=O)CNC(=O)OCc2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 2/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ACHE P22303 1/20 0.44
MMP3 P08254 3/20 0.43
HTT P42858 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
BMP1 P13497 2/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
GRK2 P25098 2/20 0.41
POLB P06746 1/20 0.41
PPARG P37231 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
NR2E3 Q9Y5X4 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
MMP2 P08253 2/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7405128 0.78 MMP1 (0.47) MMP1CA1CA2ACHEMMP3
SCHEMBL7207196 0.76 MMP13 (0.49) MMP1CA1CA2ACHEMMP3
SCHEMBL7207971 0.75 MMP13 (0.48) MMP1CA1CA2ACHEMMP3
SCHEMBL9056505 0.71 NPC1 (0.57) CA1CA2ACHEALDH1A1LMNA
Acetic Acid SCHEMBL10581041 0.70 HTT (0.60) MMP1MMP3HTTNPSR1ALDH1A1
SCHEMBL27777087 0.70 ALDH1A1 (0.58) CA1CA2HTTNPSR1ALDH1A1
SCHEMBL7862209 0.69 MMP1 (0.62) MMP1HTTNPSR1ALDH1A1LMNA
SCHEMBL11561410 0.69 NPC1 (0.65) CA1CA2ACHEHTTNPSR1
SCHEMBL27783096 0.69 NPC1 (0.65) CA1CA2ACHEHTTNPSR1
SCHEMBL8441435 0.69 ALDH1A1 (0.60) MMP1HTTALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed