SCHEMBL7405128

SCHEMBL7405128

COc1ccc(S(=O)(=O)CCC(N)SC(=O)CNC(=O)OCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 7/20 0.47
MMP13 P45452 4/20 0.47
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
ACHE P22303 2/20 0.46
ATM Q13315 1/20 0.42
MMP2 P08253 6/20 0.42
MMP3 P08254 5/20 0.42
PDE4A P27815 4/20 0.42
PDE4B Q07343 4/20 0.42
PDE4C Q08493 4/20 0.42
PDE4D Q08499 4/20 0.42
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
LMNA P02545 1/20 0.41
MMP9 P14780 1/20 0.41
BMP1 P13497 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7207972 0.78 MMP1 (0.45) MMP1MMP13CA1CA2ACHE
SCHEMBL27502837 0.76 MMP1 (0.43) MMP1MMP13MMP2MMP3PDE4A
SCHEMBL7207196 0.73 MMP13 (0.49) MMP1MMP13CA1CA2ACHE
SCHEMBL7207971 0.72 MMP13 (0.48) MMP1MMP13CA1CA2ACHE
SCHEMBL7862144 0.72 MMP13 (0.48) MMP1MMP13CA1CA2ACHE
Hydrochloric Acid SCHEMBL7862140 0.71 MMP13 (0.47) MMP1MMP13CA1CA2ACHE
SCHEMBL9056505 0.70 NPC1 (0.57) CA1CA2ACHEATMLMNA
SCHEMBL7245010 0.69 MMP2 (0.55) MMP1MMP13CA1CA2ACHE
SCHEMBL6379618 0.69 MMP2 (0.50) MMP1MMP13MMP2MMP3PDE4A
SCHEMBL7862209 0.69 MMP1 (0.62) MMP1HTTNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed