SCHEMBL7209154

SCHEMBL7209154

NC(=O)C1OCCC1(NS(=O)(=O)c1ccc(OCCc2ccc(F)cc2)cc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 17/20 0.47
MMP13 P45452 16/20 0.47
MMP2 P08253 3/20 0.42
MMP9 P14780 3/20 0.42
MMP3 P08254 2/20 0.42
MMP8 P22894 2/20 0.42
MMP14 P50281 2/20 0.42
MMP12 P39900 1/20 0.42
SGMS1 Q86VZ5 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
ADAM17 P78536 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7209180 0.92 MMP1 (0.57) MMP1MMP13MMP2MMP9MMP3
SCHEMBL25364 0.88 MMP1 (0.52) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7213095 0.84 MMP1 (0.49) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7208630 0.83 MMP13 (0.56) MMP1MMP13MMP2MMP9MMP14
SCHEMBL7208148 0.80 MMP1 (0.52) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7208607 0.78 MMP1 (0.52) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7209196 0.77 MMP1 (0.53) MMP1MMP13MMP2MMP9MMP3
SCHEMBL6953477 0.73 MMP1 (0.83) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7209150 0.72 MMP1 (0.78) MMP1MMP13MMP2MMP9MMP3
SCHEMBL7137267 0.71 MMP1 (0.59) MMP1MMP13MMP2MMP9MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
EP-1181285-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES Pfizer Products Inc. (US) 2002-02-27 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed
WO-2000073294-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PRODUCTS INC. (US) 2000-12-07 WO disclosed