SCHEMBL7208148

SCHEMBL7208148

NC(=O)C1OCCC1(NS(=O)(=O)c1ccc(Oc2ccccc2)cc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 16/20 0.52
MMP13 P45452 16/20 0.52
MMP2 P08253 5/20 0.43
MMP3 P08254 3/20 0.43
MMP9 P14780 3/20 0.43
MMP8 P22894 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
MMP14 P50281 3/20 0.43
MMP12 P39900 1/20 0.41
ADAMTS5 Q9UNA0 3/20 0.40
ADAMTS4 O75173 1/20 0.40
MEP1B Q16820 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25364 0.92 MMP1 (0.52) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7208607 0.92 MMP1 (0.52) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7209196 0.91 MMP1 (0.53) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7208630 0.87 MMP13 (0.56) MMP1MMP13MMP2MMP9MMP14
SCHEMBL7213095 0.81 MMP1 (0.49) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7209180 0.80 MMP1 (0.57) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7209154 0.80 MMP1 (0.47) MMP1MMP13MMP2MMP3MMP9
SCHEMBL2764751 0.75 ADAMTS5 (0.69) MMP1MMP13MMP2MMP3MMP9
SCHEMBL2764745 0.75 ADAMTS5 (0.69) MMP1MMP13MMP2MMP3MMP9
SCHEMBL7208592 0.72 MMP1 (0.45) MMP1MMP13MMP2MMP3MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
EP-1181285-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES Pfizer Products Inc. (US) 2002-02-27 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed
WO-2000073294-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PRODUCTS INC. (US) 2000-12-07 WO disclosed