SCHEMBL7208607

SCHEMBL7208607

NC(=O)C1OCCC1(NS(=O)(=O)c1ccc(Oc2ccc(Cl)cc2)cc1)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 17/20 0.52
MMP13 P45452 15/20 0.52
ADAMTS5 Q9UNA0 2/20 0.46
MMP9 P14780 4/20 0.43
MMP2 P08253 3/20 0.43
MMP3 P08254 3/20 0.43
MMP8 P22894 3/20 0.43
MMP14 P50281 3/20 0.43
MMP7 P09237 2/20 0.43
ADAM17 P78536 2/20 0.41
ABCB11 O95342 1/20 0.41
MMP10 P09238 1/20 0.41
PGR P06401 1/20 0.40
MMP12 P39900 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7208148 0.92 MMP1 (0.52) MMP1MMP13ADAMTS5MMP9MMP2
SCHEMBL25364 0.90 MMP1 (0.52) MMP1MMP13MMP9MMP2MMP3
SCHEMBL7209196 0.89 MMP1 (0.53) MMP1MMP13MMP9MMP2MMP3
SCHEMBL7208630 0.81 MMP13 (0.56) MMP1MMP13ADAMTS5MMP9MMP2
SCHEMBL7213095 0.80 MMP1 (0.49) MMP1MMP13ADAMTS5MMP9MMP2
SCHEMBL7209180 0.79 MMP1 (0.57) MMP1MMP13MMP9MMP2MMP3
SCHEMBL7209154 0.78 MMP1 (0.47) MMP1MMP13MMP9MMP2MMP3
Hydroxyamine SCHEMBL7514521 0.75 MMP1 (0.76) MMP1MMP13MMP9MMP2MMP3
SCHEMBL27450137 0.75 MMP1 (0.65) MMP1MMP13MMP9MMP2MMP3
SCHEMBL12076423 0.74 MMP1 (0.79) MMP1MMP13MMP9MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP claimed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US claimed
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
EP-1181285-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES Pfizer Products Inc. (US) 2002-02-27 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed
WO-2000073294-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PRODUCTS INC. (US) 2000-12-07 WO disclosed