SCHEMBL7213170

SCHEMBL7213170

O=C(Nc1ccccc1)c1cc(Br)ccc1NS(=O)(=O)c1ccc(Cl)s1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.76
KMT2A Q03164 6/20 0.76
LMNA P02545 6/20 0.76
SMN1; SMN2 Q16637 6/20 0.76
MAPT P10636 6/20 0.76
HTT P42858 6/20 0.64
RECQL P46063 3/20 0.64
ALDH1A1 P00352 3/20 0.59
POLB P06746 2/20 0.59
SLC10A6 Q3KNW5 2/20 0.59
SLC10A2 Q12908 1/20 0.59
SLC10A1 Q14973 1/20 0.59
MCOLN3 Q8TDD5 1/20 0.55
GPR27 Q9NS67 5/20 0.48
AVPR2 P30518 1/20 0.48
CCR2 P41597 1/20 0.48
GFER P55789 1/20 0.47
METAP2 P50579 1/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7120571 0.93 SMN1; SMN2 (0.65) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7214479 0.91 SLC10A6 (0.72) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7213034 0.86 MEN1 (0.57) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7208737 0.82 MEN1 (0.67) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7213183 0.81 SLC10A6 (0.73) MEN1KMT2ALMNASMN1; SMN2HTT
SCHEMBL492639 0.81 SLC10A6 (0.56) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL492766 0.79 SLC10A2 (0.52) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL492769 0.79 SLC10A2 (0.52) MEN1KMT2ALMNASMN1; SMN2MAPT
SCHEMBL7120319 0.78 SLC10A6 (0.76) MEN1KMT2ALMNASMN1; SMN2HTT
SCHEMBL27561779 0.77 SLC10A6 (0.50) MEN1KMT2ALMNASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187531-A4 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-05-28 EP claimed
US-6458845-B1 METHOD OF ANTAGONIZING A MACROPHAGE SCAVENGER RECEPTOR COMPRISING ADMINISTERING TO A SUBJECT IN NEED OF TREATMENT AN EFFECTIVE AMOUNT OF AN N-PHENYL-2-(3-TRIFLUOROMETHYLPHENYLSULFONAMIDO)BENZAMIDE, A SMITHKLINE BEECHAM CORPORATION 2002-10-01 US claimed
EP-1187531-A1 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-03-20 EP claimed
WO-2001098264-A1 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-27 WO claimed
WO-2000078145-A1 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-28 WO claimed
EP-1187531-A4 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-05-28 EP disclosed
US-6458845-B1 METHOD OF ANTAGONIZING A MACROPHAGE SCAVENGER RECEPTOR COMPRISING ADMINISTERING TO A SUBJECT IN NEED OF TREATMENT AN EFFECTIVE AMOUNT OF AN N-PHENYL-2-(3-TRIFLUOROMETHYLPHENYLSULFONAMIDO)BENZAMIDE, A SMITHKLINE BEECHAM CORPORATION 2002-10-01 US disclosed
EP-1187531-A1 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-03-20 EP disclosed
WO-2001098264-A1 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-27 WO disclosed
WO-2000078145-A1 MACROPHAGE SCAVENGER RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2000-12-28 WO disclosed