SCHEMBL7214293

SCHEMBL7214293

CCOC(=O)Cn1c(C)cc(C#Cc2ccccc2)cc1=O

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.53
RAB9A P51151 1/20 0.53
ALDH1A1 P00352 3/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
TSHR P16473 3/20 0.48
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7214686 0.78 ALDH1A1 (0.56) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL7214682 0.78 ALDH1A1 (0.56) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL7214687 0.78 ALDH1A1 (0.56) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL2828050 0.76 KDM4E (0.54) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL7220336 0.75 POLB (0.62) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL2827984 0.73 ALDH1A1 (0.59) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL11277508 0.73 KDM4E (0.58) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL7216109 0.72 SMN1; SMN2 (0.49) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL7216097 0.72 SMN1; SMN2 (0.49) KDM4ERAB9AALDH1A1MEN1KMT2A
SCHEMBL7216103 0.72 SMN1; SMN2 (0.49) KDM4ERAB9AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610692-B1 Anticoagulants MERCK & CO., INC. 2003-08-26 US disclosed
EP-1124822-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2002-04-03 EP disclosed
EP-1124822-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2001-08-22 EP disclosed
WO-2000026211-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2000-05-11 WO disclosed