SCHEMBL7214768

SCHEMBL7214768

CC#Cc1cnc2ccccc2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
CYP1A2 P05177 2/20 0.53
PARP1 P09874 1/20 0.50
CYP1A1 P04798 1/20 0.47
CYP1B1 Q16678 1/20 0.47
ACACB O00763 1/20 0.47
PDGFRB P09619 3/20 0.46
PDGFRA P16234 3/20 0.46
MGAM O43451 1/20 0.43
PIK3CA P42336 2/20 0.42
PIK3CD O00329 1/20 0.42
EGFR P00533 1/20 0.42
HTR3A P46098 1/20 0.41
MTOR P42345 1/20 0.41
CYP2A6 P11509 1/20 0.41
BIRC5 O15392 1/20 0.40
GLA P06280 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18253193 0.84 ALDH1A1 (0.58) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL18253192 0.83 ALDH1A1 (0.65) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL27614825 0.82 ALDH1A1 (0.59) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL547195 0.82 ALDH1A1 (0.59) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL4818276 0.81 ALDH1A1 (0.63) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL15112998 0.81 ALDH1A1 (0.58) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL10162702 0.81 ALDH1A1 (0.71) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL3061440 0.81 ALDH1A1 (0.58) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL11300052 0.78 ALDH1A1 (0.55) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA
SCHEMBL23781564 0.77 ALDH1A1 (0.71) ALDH1A1CYP1A2ACACBPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1373767-A Ketolide antibacterials ORTHO MCNEIL PHARM INC (US) 2002-10-09 CN claimed
EP-1506214-B1 6-11 BICYCLIC KETOLIDE DERIVATIVES ENANTA PHARM INC (US) 2010-01-20 EP disclosed
EP-1272500-A2 PROCESS FOR PREPARING 6-O-ALKENYL-SUBSITUTED ERYTHROMYCIN DERIVATIVES Abbott Laboratories (US) 2003-01-08 EP disclosed
EP-1192139-A1 PREPARATION OF QUINOLINE-SUBSTITUTED CARBONATE AND CARBAMATE DERIVATIVES Abbott Laboratories (US) 2002-04-03 EP disclosed
WO-2001000582-A1 PREPARATION OF QUINOLINE-SUBSTITUTED CARBONATE AND CARBAMATE DERIVATIVES ABBOTT LABORATORIES (US) 2001-01-04 WO disclosed
WO-2000078773-A2 PROCESS FOR PREPARING 6-O-ALKENYL-SUBSTITUTED ERYTHROMYCIN DERIV ATIVES ABBOTT LABORATORIES (US) 2000-12-28 WO disclosed