SCHEMBL7215162

SCHEMBL7215162

OCCCNc1cccc(F)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.54
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
KCNH3 Q9ULD8 4/20 0.48
ALDH1A1 P00352 3/20 0.47
HPGD P15428 1/20 0.46
HTT P42858 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 2/20 0.43
IDO1 P14902 1/20 0.43
EGFR P00533 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7214593 0.94 ALDH1A1 (0.54) KDRMEN1KMT2AKCNH3ALDH1A1
SCHEMBL1431624 0.88 MEN1 (0.53) KDRMEN1KMT2AKCNH3ALDH1A1
SCHEMBL11119734 0.82 ALDH1A1 (0.68) MEN1KMT2AALDH1A1HPGDHTT
SCHEMBL12355294 0.82 MEN1 (0.55) MEN1KMT2AALDH1A1HPGDHTT
SCHEMBL11115860 0.81 HPGD (0.46) KDRMEN1KMT2AALDH1A1HPGD
SCHEMBL7214532 0.81 MAPT (0.47) MEN1KMT2AALDH1A1HPGDHTT
SCHEMBL5159176 0.81 HTR7 (0.51) MEN1KMT2AKCNH3ALDH1A1HTT
SCHEMBL4155729 0.81 MEN1 (0.50) MEN1KMT2AALDH1A1HPGDHTT
SCHEMBL27642277 0.81 F2R (0.48) MEN1KMT2AALDH1A1HPGDHTT
SCHEMBL5541987 0.81 HPGD (0.46) KDRMEN1KMT2AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6630485-B2 For therapy of inflammatory disease SYNTEX (U.S.A.) LLC 2003-10-07 US disclosed
US-6316464-B1 P38 MAP kinase inhibitors SYNTEX (U.S.A.) LLC 2001-11-13 US disclosed
EP-0058868-B1 DERIVATIVES OF TETRAHYDROPYRIMIDINON, PROCESS FOR THEIR PREPARATION AND HERBICIDES CONTAINING THOSE DERIVATIVES AS ACTIVE PRODUCTS NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1984-04-11 EP disclosed
US-4402731-A Herbicidally active novel substituted tetrahydropyrimidinones NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1983-09-06 US disclosed
EP-0058868-A1 Derivatives of tetrahydropyrimidinon, process for their preparation and herbicides containing those derivatives as active products NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1982-09-01 EP disclosed