SCHEMBL7216396

SCHEMBL7216396

O=C(O)C1=Cc2cc(C#Cc3ccccc3)ccc2OCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.51
ACACB O00763 4/20 0.43
HNF4A P41235 1/20 0.41
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
DRD1 P21728 1/20 0.38
DRD5 P21918 1/20 0.38
OPRM1 P35372 1/20 0.38
P2RY6 Q15077 1/20 0.38
S1PR5 Q9H228 2/20 0.37
ALOX5 P09917 1/20 0.37
FFAR1 O14842 3/20 0.36
PTPN11 Q06124 1/20 0.34
CYP26A1 O43174 1/20 0.34
CYP3A4 P08684 1/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
CRABP2 P29373 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218118 0.87 GRM5 (0.46) GRM5ACACBP2RY6ALOX5
SCHEMBL5208747 0.84 PTGS2 (0.48) ACACBP2RY6ALOX5
SCHEMBL913383 0.78 ALOX5 (0.49) ALOX5
SCHEMBL6755749 0.77 ALOX5 (0.43) ALOX5
SCHEMBL6755727 0.76 CA12 (0.46)
SCHEMBL6756847 0.76 MEN1 (0.37) P2RY6ALOX5
SCHEMBL6756803 0.76 MEN1 (0.52)
SCHEMBL7677996 0.73 CCR5 (0.43) ALOX5
SCHEMBL6756877 0.73 MTNR1A (0.52) ALOX5
SCHEMBL5208620 0.72 CCR5 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed