SCHEMBL7216713

SCHEMBL7216713

CCN(CC)c1ccc(N)cc1.Nc1ncnc2nn[nH]c12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.50
ALDH1A1 P00352 2/20 0.50
PSMD14 O00487 1/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
MAPK1 P28482 1/20 0.50
RECQL P46063 1/20 0.50
GFER P55789 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
LMNA P02545 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MAPT P10636 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PIK3CD O00329 2/20 0.36
PIK3CA P42336 2/20 0.36
PIK3CB P42338 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216711 0.80 ALDH1A1 (0.51) TDP1ALDH1A1PSMD14CYP3A4TSHR
SCHEMBL29471407 0.78 PI4KA (0.50) TSHRLMNAPIK3CDPIK3CAPIK3CB
SCHEMBL24640 0.78 PI4KA (0.50) TSHRLMNAPIK3CDPIK3CAPIK3CB
Ammonia Solution, Strong SCHEMBL28104176 0.76 PI4KA (0.48) TSHRLMNAPIK3CDPIK3CAPIK3CB
Benzene SCHEMBL28791218 0.75 PI4KA (0.47) ALDH1A1LMNAPIK3CDPIK3CAPIK3CB
SCHEMBL8467252 0.71 ALDH1A1 (1.00) TDP1ALDH1A1PSMD14CYP3A4TSHR
SCHEMBL33781 0.71 ALDH1A1 (1.00) TDP1ALDH1A1PSMD14CYP3A4TSHR
Iodide SCHEMBL5069469 0.69 ALDH1A1 (0.86) TDP1ALDH1A1PSMD14CYP3A4TSHR
Hydrochloric Acid SCHEMBL970320 0.69 ALDH1A1 (0.95) TDP1ALDH1A1PSMD14CYP3A4TSHR
Hydrochloric Acid SCHEMBL970321 0.69 ALDH1A1 (0.95) TDP1ALDH1A1PSMD14CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339702-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2003-09-03 EP disclosed
WO-2001068619-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEX INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-09-20 WO disclosed