SCHEMBL7217060

SCHEMBL7217060

COc1ccc(C(=O)Cc2ccc(S(N)(=O)=O)cc2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.52
PTGS2 P35354 4/20 0.52
CA1 P00915 5/20 0.52
CA2 P00918 5/20 0.52
CA9 Q16790 5/20 0.52
CA7 P43166 1/20 0.52
CA14 Q9ULX7 1/20 0.52
TSHR P16473 1/20 0.52
NLRP3 Q96P20 1/20 0.49
ALDH1A1 P00352 3/20 0.48
CA12 O43570 2/20 0.48
CA4 P22748 1/20 0.47
NPC1 O15118 1/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
USP2 O75604 1/20 0.46
PDE4D Q08499 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170001 0.85 PTGS2 (0.53) PTGS1PTGS2CA1CA2CA9
SCHEMBL7220907 0.81 MAPT (0.55) ALDH1A1NPC1LMNAHTTMEN1
SCHEMBL6170212 0.80 LMNA (0.49) ALDH1A1NPC1LMNAHTTMEN1
SCHEMBL6168504 0.79 CA2 (0.65) CA1CA2CA9CA7CA14
SCHEMBL22516210 0.78 CA1 (0.65) CA1CA2CA9CA7ALDH1A1
SCHEMBL2315314 0.76 PTGS2 (0.66) PTGS1PTGS2CA1CA2CA9
SCHEMBL7214644 0.76 PTGS2 (0.53) PTGS1PTGS2CA1CA2CA9
SCHEMBL22570710 0.75 TAS1R3 (0.51) TSHRALDH1A1NPC1LMNAHTT
SCHEMBL6168486 0.74 CA1 (0.62) CA1CA2CA9CA7ALDH1A1
Hydrochloric Acid SCHEMBL29393777 0.74 TAS1R3 (0.50) TSHRALDH1A1NPC1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6670365-B1 Treatment of inflamation and/or cyclooxygenase-mediated diseases, reduced ulcerogenic effects; 2-phenyl-3-(4-methylsulfonylphenyl)imidazo(1,2-a)pyrimidine LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2003-12-30 US disclosed
EP-1104762-B1 SUBSTITUTED IMIDAZO[1,2A]AZINES AS SELECTIVE INHIBITORS OF COX-2 S A L V A T LAB SA (ES) 2002-09-18 EP disclosed
EP-1104762-A1 SUBSTITUTED IMIDAZO 1,2A]AZINES AS SELECTIVE INHIBOTORS OF COX-2 LABORATORIOS S.A.L.V.A.T., S.A. (ES) 2001-06-06 EP disclosed