SCHEMBL7217403

SCHEMBL7217403

C/C(=C/c1ccccc1)C1CCc2ccccc2O1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 5/20 0.46
HSD11B1 P28845 1/20 0.41
AOC2 O75106 5/20 0.40
MAOA P21397 5/20 0.40
MAOB P27338 5/20 0.40
DAO P14920 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
CYP2D6 P10635 2/20 0.38
OPRK1 P41145 2/20 0.38
CA2 P00918 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7217412 1.00 KDM1A (0.46) KDM1AHSD11B1AOC2MAOAMAOB
SCHEMBL7217406 0.78 HSD11B1 (0.41) HSD11B1AOC2MAOAMAOBDAO
SCHEMBL12060986 0.76 HSD11B1 (0.42) HSD11B1AOC2MAOAMAOBDAO
SCHEMBL8039734 0.76 HSD11B1 (0.47) HSD11B1HDAC3HDAC1HDAC2CYP2D6
SCHEMBL4934593 0.74 HDAC3 (0.49) HSD11B1AOC2MAOAMAOBDAO
SCHEMBL229558 0.74 HPGD (0.49) HSD11B1HDAC3HDAC1HDAC2CYP2D6
SCHEMBL30887999 0.74 HDAC3 (0.49) HSD11B1AOC2MAOAMAOBDAO
SCHEMBL2286036 0.74 HPGD (0.49) HSD11B1HDAC3HDAC1HDAC2CYP2D6
SCHEMBL5695491 0.74 HDAC3 (0.49) HSD11B1AOC2MAOAMAOBDAO
SCHEMBL430259 0.74 HDAC3 (0.49) HSD11B1AOC2MAOAMAOBDAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627652-B1 Treatment of diseases or conditions of the type which are normally treated with retinoid-like compounds is disclosed, with pharmaceutical compositions containing an active compound which is a selective agonist of the RXR retinoid ALLERGAN, INC. 2003-09-30 US disclosed
US-6624188-B1 Administered to treat or prevent one or more of the diseases and conditions selected from the group consisting of dermatoses, atherosclerosis and restenosis resulting from neointimal hyperproliferation, non-malignant and ALLERGAN, INC. 2003-09-23 US disclosed
US-5455265-A For mammals; skin disorders, cancer, inflammatory disease, cardiovascular diorders, autoimmune diseases and others ALLERGAN, INC. (US) 1995-10-03 US disclosed
US-5324840-A Skin disorders ALLERGAN, INC. (US) 1994-06-28 US disclosed