SCHEMBL7217586

SCHEMBL7217586

CC(=Cc1ccc(C)cc1)c1ccc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTGS1 P23219 2/20 0.46
PTGS2 P35354 2/20 0.46
NQO2 P16083 1/20 0.46
ESR1 P03372 1/20 0.46
ESR2 Q92731 1/20 0.46
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7217591 0.90 CYP2A6 (0.47) CYP2A6TDP1PTGS1PTGS2NQO2
SCHEMBL7217583 0.90 CYP2A6 (0.47) CYP2A6TDP1PTGS1PTGS2NQO2
SCHEMBL9806282 0.88 CYP1B1 (0.51) TDP1PTGS1PTGS2NQO2ESR1
SCHEMBL9806279 0.88 CYP1B1 (0.51) TDP1PTGS1PTGS2NQO2ESR1
SCHEMBL18790028 0.80 ESR1 (0.68) CYP2A6TDP1PTGS1PTGS2NQO2
SCHEMBL6546605 0.80 ESR1 (0.68) CYP2A6TDP1PTGS1PTGS2NQO2
SCHEMBL4602278 0.78 MAPT (0.59) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL6547576 0.78 ESR1 (0.55) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL7570852 0.76 CES2 (0.54) TDP1CES2CES1MAPTKDM4E
SCHEMBL28539564 0.76 CES2 (0.54) TDP1CES2CES1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627652-B1 Treatment of diseases or conditions of the type which are normally treated with retinoid-like compounds is disclosed, with pharmaceutical compositions containing an active compound which is a selective agonist of the RXR retinoid ALLERGAN, INC. 2003-09-30 US disclosed
US-6624188-B1 Administered to treat or prevent one or more of the diseases and conditions selected from the group consisting of dermatoses, atherosclerosis and restenosis resulting from neointimal hyperproliferation, non-malignant and ALLERGAN, INC. 2003-09-23 US disclosed
US-5455265-A For mammals; skin disorders, cancer, inflammatory disease, cardiovascular diorders, autoimmune diseases and others ALLERGAN, INC. (US) 1995-10-03 US disclosed
US-5324840-A Skin disorders ALLERGAN, INC. (US) 1994-06-28 US disclosed