SCHEMBL7217804

SCHEMBL7217804

COc1ccc(CC(C)OC2CCCCO2)c(CBr)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HTR2A P28223 1/20 0.35
TSHR P16473 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTT P42858 1/20 0.33
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7212889 0.85 KDM4E (0.33) NPC1RAB9ATSHRKDM4EALDH1A1
SCHEMBL7211776 0.82 KDM4C (0.36) NPC1RAB9AHTR2AMEN1KMT2A
SCHEMBL9123646 0.76 DHFR (0.35) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL9119549 0.76 DHFR (0.31)
SCHEMBL2014844 0.75 ALDH1A1 (0.36) MEN1KMT2AALDH1A1MAPTLMNA
SCHEMBL7050550 0.72 SIGMAR1 (0.39) MEN1KMT2A
SCHEMBL6400656 0.72 NPC1 (0.50) NPC1RAB9AMEN1KMT2A
SCHEMBL17145065 0.72 DPP4 (0.41) HTR2A
SCHEMBL16543024 0.71 NPC1 (0.41) NPC1RAB9ATSHRALDH1A1GAA
SCHEMBL6253588 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178960-B1 VITAMIN D ANALOGUES AND THEIR PHARMACEUTICAL USE LEO PHARMA AS (DK) 2003-11-05 EP disclosed
EP-1178960-A1 VITAMIN D ANALOGUES AND THEIR PHARMACEUTICAL USE LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 2002-02-13 EP disclosed
WO-2000064869-A1 VITAMIN D ANALOGUES AND THEIR PHARMACEUTICAL USE Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 2000-11-02 WO disclosed