SCHEMBL7218366

SCHEMBL7218366

CC(=NO)NCCCC(N)C(=O)c1ncc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
HSPA5 P11021 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
DPP7 Q9UHL4 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218361 1.00 NPC1 (0.33) NPC1RAB9AHSPA5MEN1KMT2A
SCHEMBL7218372 0.80 NOS1 (0.37) NPC1RAB9AMEN1KMT2A
SCHEMBL28044670 0.76 GSR (0.43) NPC1RAB9AKMT2ADPP7
SCHEMBL7611110 0.70 NPY4R (0.43)
SCHEMBL7172385 0.68 NOS2 (0.50) MEN1KMT2ADPP7
SCHEMBL7915399 0.68 NOS2 (0.50) MEN1KMT2ADPP7
SCHEMBL28612372 0.67 NPC1 (0.46) NPC1RAB9AHSPA5KMT2AKDM4E
SCHEMBL11599997 0.67 NPC1 (0.46) NPC1RAB9AHSPA5KMT2AKDM4E
Hydrochloric Acid SCHEMBL7218895 0.67 NOS2 (0.51) MEN1KMT2ADPP7
SCHEMBL7227260 0.67 DPP7 (0.42) MEN1KMT2ADPP7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6576780-B1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors GD SEARLE & COMPANY 2003-06-10 US claimed
US-6576780-B1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors GD SEARLE & COMPANY 2003-06-10 US disclosed
US-6207708-B1 FOR THERAPY AND PROPHYLAXIS OF AUTOIMMUNE AND/OR INFLAMMATORY CONDITIONS AFFECTING THE JOINTS SUCH AS ARTHRITIS, AND INFLAMMATORY BOWEL DISEASE, CARDIVASCULAR ISCHEMIA, DIABETES, CONGESTIVE HEART FAILURE, MYOCARDITIS, ATHEROSCLEROSIS, G. D. SEARLE & COMPANY 2001-03-27 US disclosed