SCHEMBL7218429

SCHEMBL7218429

CCOC(=O)Oc1c[nH]c2cc([N+](=O)[O-])c(F)cc2c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
HPGD P15428 2/20 0.39
TP53 P04637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
GABRA1 P14867 3/20 0.38
GABRB2 P47870 3/20 0.38
GABRB1 P18505 2/20 0.38
GABRA3 P34903 2/20 0.38
MAPT P10636 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 2/20 0.35
GALR2 O43603 1/20 0.34
MITF O75030 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4840379 0.84 GABRA1 (0.56) ALDH1A1MEN1KMT2AHPGDTP53
SCHEMBL8556198 0.80 MEN1 (0.39) MTNR1AMTNR1BALDH1A1MEN1KMT2A
SCHEMBL810412 0.77 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AHPGDL3MBTL1
SCHEMBL7219604 0.76 NQO2 (0.41) NQO2MTNR1AMTNR1BALDH1A1MEN1
SCHEMBL18306134 0.74 CUL4A (0.45) ALDH1A1MEN1KMT2AHPGDMAPT
SCHEMBL31047098 0.74 CUL4A (0.45) ALDH1A1MEN1KMT2AHPGDL3MBTL1
SCHEMBL810673 0.74 CUL4A (0.45) ALDH1A1MEN1KMT2AHPGDL3MBTL1
SCHEMBL4306866 0.74 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AHPGDHSD17B10
SCHEMBL9491783 0.72 HTR2B (0.43) MTNR1AMTNR1BALDH1A1HPGDHSD17B10
SCHEMBL8367665 0.71 ALDH1A1 (0.43) ALDH1A1MEN1KMT2AHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362034-A1 QUINOLINE, ISOQUINOLINE AND PHTHALAZINE DERIVATIVES AS ANTAGONISTS OF THE GONADOTROPIN-RELEASING HORMONE Schering Aktiengesellschaft (DE) 2003-11-19 EP disclosed
WO-2002066437-A1 QUINOLINE, ISOQUINOLINE AND PHTHALAZINE DERIVATIVES AS ANTAGONISTS OF THE GONADOTROPIN-RELEASING HORMONE ZENTARIS GMBH (DE) 2002-08-29 WO disclosed