SCHEMBL7219604

SCHEMBL7219604

CCOC(=O)Oc1c[nH]c2ccc(F)c([N+](=O)[O-])c2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.41
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GABRA1 P14867 3/20 0.36
GABRB2 P47870 3/20 0.36
GABRB1 P18505 2/20 0.35
GABRA3 P34903 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4835712 0.82 GABRA1 (0.50) KMT2AALDH1A1MEN1TP53HPGD
SCHEMBL7218429 0.76 NQO2 (0.40) NQO2MTNR1AMTNR1BKMT2AALDH1A1
SCHEMBL3837986 0.71 KMT2A (0.41) KMT2AALDH1A1MEN1TP53HPGD
SCHEMBL3842038 0.71 GABRA1 (0.39) KMT2AALDH1A1MEN1TP53HPGD
SCHEMBL3839419 0.70 MEN1 (0.37) KMT2AALDH1A1MEN1TP53HPGD
SCHEMBL3837988 0.69 HSD17B10 (0.39) MTNR1AMTNR1BKMT2AALDH1A1MEN1
SCHEMBL3250627 0.67 MAPT (0.46) NQO2KMT2AALDH1A1MEN1
SCHEMBL8556198 0.65 MEN1 (0.39) MTNR1AMTNR1BKMT2AALDH1A1MEN1
SCHEMBL810412 0.65 ALDH1A1 (0.43) KMT2AALDH1A1MEN1HPGDL3MBTL1
SCHEMBL28857890 0.65 RAB9A (0.51) KMT2AALDH1A1MEN1L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362034-A1 QUINOLINE, ISOQUINOLINE AND PHTHALAZINE DERIVATIVES AS ANTAGONISTS OF THE GONADOTROPIN-RELEASING HORMONE Schering Aktiengesellschaft (DE) 2003-11-19 EP disclosed
WO-2002066437-A1 QUINOLINE, ISOQUINOLINE AND PHTHALAZINE DERIVATIVES AS ANTAGONISTS OF THE GONADOTROPIN-RELEASING HORMONE ZENTARIS GMBH (DE) 2002-08-29 WO disclosed