SCHEMBL7219562

SCHEMBL7219562

CCOCn1cc(/C=C/Br)c(=O)[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TK2 O00142 6/20 0.41
TK1 P04183 3/20 0.41
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
UPP1 Q16831 1/20 0.36
MAPK1 P28482 1/20 0.34
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7219565 1.00 TK2 (0.41) TK2TK1CYP1A2CYP3A4TSHR
SCHEMBL23981077 0.77 TK1 (0.35) TK2TK1CYP1A2CYP3A4TSHR
SCHEMBL7213283 0.76 KMT2A (0.48) TK1CYP1A2BLMUPP1MAPK1
SCHEMBL1558433 0.76 TK2 (0.42) TK2TK1CYP1A2CYP3A4TSHR
SCHEMBL1558432 0.76 TK2 (0.42) TK2TK1CYP1A2CYP3A4TSHR
SCHEMBL7213472 0.74 UPP1 (0.47) TK1UPP1MAPK1
SCHEMBL7219926 0.74 MAPK1 (0.54) TK2TK1NPSR1MAPK1HPGD
SCHEMBL2180462 0.73 HPGD (0.60) TK2MAPK1HPGD
SCHEMBL1558585 0.73 HPGD (0.60) TK2MAPK1HPGD
SCHEMBL6372044 0.73 LMNA (0.56) CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37979-E1 Pyrimidine derivatives and anti-viral agent containing the same as active ingredient thereof MITSUBISHI CHEMICAL CORPORATION 2003-02-04 US disclosed
US-5461060-A Antiretroviral activity MITSUBISHI KASEI CORPORATION (JP) 1995-10-24 US disclosed
EP-0420763-A2 6-Substituted acyclopyrimidine nucleoside derivatives and antiviral agent containing the same as active ingredient thereof Mitsubishi Chemical Corporation (JP) 1991-04-03 EP disclosed