SCHEMBL721964

SCHEMBL721964

NC(=S)Nc1ccc2[nH]ccc2c1

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOB P27338 11/20 0.65
MAOA P21397 10/20 0.65
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
MAPT P10636 3/20 0.56
PRKCI P41743 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4518907 0.86 ESR1 (0.52) MAOBMAOANPC1RAB9AMAPT
SCHEMBL31668680 0.84 MAOB (0.88) MAOBMAOANPC1RAB9AMAPT
SCHEMBL4526884 0.83 MAOB (0.65) MAOBMAOANPC1RAB9AMAPT
SCHEMBL1576877 0.83 NPC1 (0.63) MAOBMAOANPC1RAB9AMAPT
SCHEMBL9540720 0.83 F2 (0.57) MAOBMAOANPC1RAB9AMAPT
SCHEMBL30026512 0.83 NPC1 (0.63) MAOBMAOANPC1RAB9AMAPT
SCHEMBL22803696 0.79 NPC1 (0.67) MAOBMAOANPC1RAB9AMAPT
SCHEMBL4347943 0.77 NPC1 (0.69) MAOBMAOANPC1RAB9AMAPT
SCHEMBL31668688 0.77 MAOA (0.66) MAOBMAOANPC1RAB9AMAPT
SCHEMBL5177372 0.76 MAOB (0.83) MAOBMAOANPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 64 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250188072-A1 COMPOUNDS FOR TREATMENT OF CANCER UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2025-06-12 US disclosed
US-12187720-B2 Compounds for treatment of cancer UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2025-01-07 US disclosed
CN-111253336-B Compounds for the treatment of cancer GTX公司 2023-11-21 CN disclosed
US-11465987-B2 Compounds for treatment of cancer Oncternal Therapeutics, Inc. (US) 2022-10-11 US disclosed
US-20220024912-A1 COMPOUNDS FOR TREATMENT OF CANCER Oncternal Therapeutics, Inc. (US) 2022-01-27 US disclosed
US-11084811-B2 Compounds for treatment of cancer Oncternal Therapeutics, Inc. (US) 2021-08-10 US disclosed
CN-106794174-B Compounds for the treatment of cancer GTX公司 2021-03-12 CN disclosed
EP-3708164-A1 COMPOUNDS FOR TREATMENT OF CANCER Oncternal Therapeutics, Inc (US) 2020-09-16 EP disclosed
CN-111253336-A Compounds for the treatment of cancer GTX公司 2020-06-09 CN disclosed
EP-3139919-B1 COMPOUNDS FOR TREATMENT OF CANCER ONCTERNAL THERAPEUTICS INC (US) 2020-06-03 EP disclosed
EP-1883451-A2 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY Neuraxon Inc. (CA) 2008-02-06 EP disclosed
WO-2007063418-A2 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2007-06-07 WO disclosed
WO-2007063418-A2 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON, INC. (CA) 2007-06-07 WO disclosed
WO-2007042321-A2 KINASE INHIBITORS DEVGEN N.V. (BE) 2007-04-19 WO disclosed
US-20060258721-A1 Substituted indole compounds having NOS inhibitory activity NEURAXON INC. (CA) 2006-11-16 US disclosed
EP-0619805-B1 5-(HETERO- OR CARBOCYCLYLAMINO)-INDOLE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS 5-HT1 AGONISTS PFIZER (US) 2000-03-15 EP disclosed
CN-1045294-C Indole derivatives PFIZER (US) 1999-09-29 CN disclosed
US-5639752-A SEROTONIN AGONIST PFIZER INC (US) 1997-06-17 US disclosed
EP-0619805-A1 INDOLE DERIVATIVES PFIZER HOSPITAL PRODUCTS, INC. (US) 1994-10-19 EP disclosed
WO-1993011106-A1 INDOLE DERIVATIVES PFIZER, INC. (US) 1993-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12187720-B2 Compounds for treatment of cancer KLK3, BRDT, ACP3 MAOB 2022/4885MAOA 2964/4885NPC1 1453/4885
US-11084811-B2 Compounds for treatment of cancer KLK3, BRDT, ACP3 MAOB 2022/4885MAOA 2964/4885NPC1 1453/4885
US-20220024912-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 MAOB 2022/4885MAOA 2964/4885NPC1 1453/4885
US-20060258721-A1 Substituted indole compounds having NOS inhibitory activity NOS2, NOS1, NOS3 MAOB 36/4885MAOA 19/4885NPC1 906/4885
US-20250188072-A1 COMPOUNDS FOR TREATMENT OF CANCER KLK3, BRDT, ACP3 MAOB 2022/4885MAOA 2964/4885NPC1 1453/4885
US-11465987-B2 Compounds for treatment of cancer KLK3, BRDT, ACP3 MAOB 2022/4885MAOA 2964/4885NPC1 1453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.