SCHEMBL7220708

SCHEMBL7220708

Cc1nc(C)c(-c2cscn2)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.53
HTT P42858 1/20 0.53
CDK4 P11802 4/20 0.49
CDK2 P24941 4/20 0.49
CCNE1 P24864 1/20 0.49
TRPV4 Q9HBA0 5/20 0.45
COMT P21964 2/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43
TUBA1C Q9BQE3 1/20 0.43
TUBB6 Q9BUF5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16434004 0.72 LMNA (0.72) LMNAHTTTRPV4TUBB4ATUBB
SCHEMBL3799747 0.72 ALDH1A1 (0.43) LMNAHTTNPC1MEN1KMT2A
SCHEMBL12537263 0.71 COMT (0.52) LMNAHTTCDK4CDK2CCNE1
SCHEMBL16434062 0.69 LMNA (1.00) LMNAHTTCDK4CDK2CCNE1
SCHEMBL7964249 0.68 TSHR (0.50) NPC1METAP1RAB9AALDH1A1TSHR
SCHEMBL9286689 0.68 ALDH1A1 (0.43) HTTNPC1METAP1RAB9APOLB
SCHEMBL5352893 0.66 CDK2 (0.45) LMNAHTTCDK4CDK2CCNE1
SCHEMBL4314069 0.66 CDK2 (1.00) LMNAHTTCDK4CDK2CCNE1
SCHEMBL12912141 0.66 TRPV4 (0.64) LMNAHTTTRPV4TUBB4ATUBB
SCHEMBL5209668 0.65 LMNA (0.49) LMNAHTTCDK4CDK2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3344997-A1 OPIOID RECEPTOR MODULATORS AND USE THEREOF Regents of the University of Minnesota (US) 2018-07-11 EP disclosed
WO-2017039778-A1 OPIOID RECEPTOR MODULATORS AND USE THEREOF REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2017-03-09 WO disclosed
US-6605631-B1 Controlling fungi and pests; improved activity and plant tolerability BASF AKTIENGESELLSCHAFT (DE) 2003-08-12 US disclosed