SCHEMBL7224289

SCHEMBL7224289

Cc1ccc(-c2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)o1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 10/20 0.36
HTR3E A5X5Y0 5/20 0.36
HTR3B O95264 5/20 0.36
HTR3A P46098 5/20 0.36
HTR3D Q70Z44 5/20 0.36
HTR3C Q8WXA8 5/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ESR1 P03372 1/20 0.34
ESRRG P62508 1/20 0.34
ESR2 Q92731 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPN11 Q06124 1/20 0.34
SMYD3 Q9H7B4 1/20 0.34
AKT1 P31749 1/20 0.34
SLC6A2 P23975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7232161 0.89 CHRNA7 (0.38) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7230457 0.87 CHRNA7 (0.37) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7233633 0.85 ITK (0.39) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224299 0.83 NPC1 (0.45) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7225477 0.82 CHRNA7 (0.36) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7224991 0.81 ESRRG (0.46) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7233692 0.81 TXK (0.36) CHRNA7HTR3EHTR3BHTR3AHTR3D
SCHEMBL7223510 0.81 NPC1 (0.52) CHRNA7NPC1RAB9ASLC6A2SLC6A4
SCHEMBL7224346 0.81 SLC6A3 (0.33) NPC1RAB9ATP53HPGDTSHR
SCHEMBL7233342 0.81 NPC1 (0.33) NPC1RAB9ATP53HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed