SCHEMBL7224671

SCHEMBL7224671

Cn1c(CCc2ccc(CN)cc2)nc2cc(N(Cc3cccc4ccccc34)C(=O)CN3CCC(Nc4ccccc4Cl)CC3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 7/20 0.40
NTRK2 Q16620 7/20 0.40
F2 P00734 2/20 0.37
HDAC1 Q13547 2/20 0.35
KCNH2 Q12809 2/20 0.35
MCHR1 Q99705 2/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
DRD4 P21917 1/20 0.34
ROCK2 O75116 1/20 0.34
CCR2 P41597 1/20 0.34
ROCK1 Q13464 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7115891 0.94 F2 (0.46) NTRK1NTRK2F2HDAC1HDAC6
SCHEMBL7218890 0.91 NTRK1 (0.40) NTRK1NTRK2F2KCNH2MCHR1
SCHEMBL7222786 0.90 NTRK1 (0.44) NTRK1NTRK2F2HDAC1KCNH2
SCHEMBL7219016 0.89 CA12 (0.41) NTRK1NTRK2F2HDAC1KDM4E
SCHEMBL7223673 0.89 F2 (0.39) NTRK1NTRK2F2HDAC1KCNH2
SCHEMBL7216788 0.89 KDM4E (0.39) NTRK1NTRK2F2HDAC1KCNH2
SCHEMBL7223705 0.88 NTRK1 (0.45) NTRK1NTRK2F2HDAC1KDM4E
SCHEMBL7216888 0.87 F2 (0.37) NTRK1NTRK2F2HDAC1KDM4E
SCHEMBL7217499 0.86 F2 (0.42) F2HDAC1KCNH2KDM4ENPC1
SCHEMBL7219009 0.85 F2 (0.41) F2HDAC1KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6656956-B2 Tryptase inhibitor; antiinflamamtory agents, antiallergens BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-12-02 US disclosed