SCHEMBL7224696

SCHEMBL7224696

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(Sc2ccc(Cl)c(Cl)c2)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.40
SLC6A4 P31645 5/20 0.40
CHRNB2 P17787 6/20 0.35
CHRNA4 P43681 6/20 0.35
SLC6A2 P23975 3/20 0.35
CHRNB4 P30926 3/20 0.35
CHRNA3 P32297 3/20 0.35
CHRNA1 P02708 2/20 0.35
CHRNG P07510 2/20 0.35
CHRNB1 P11230 2/20 0.35
CHRND Q07001 2/20 0.35
ITGA5 P08648 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.31
TAS1R2 Q8TE23 1/20 0.31
CHRNA7 P36544 4/20 0.31
ALDH1A1 P00352 2/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
HPGD P15428 1/20 0.31
CHRNA2 Q15822 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231748 0.89 SLC6A4 (0.39) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2
SCHEMBL7224680 0.88 CHRNB2 (0.36) SLC6A3SLC6A4CHRNB2CHRNA4
SCHEMBL7226264 0.87 SLC6A3 (0.33) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2
SCHEMBL7223814 0.87 SLC6A3 (0.33) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2
SCHEMBL7225963 0.85 SLC6A3 (0.39) SLC6A3SLC6A4SLC6A2
SCHEMBL7226364 0.85 HTR3E (0.35) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2
SCHEMBL7232697 0.84 KDM4C (0.35) SLC6A3CHRNB2CHRNA4ALDH1A1
SCHEMBL7230561 0.84 ITGB2 (0.35) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2
SCHEMBL7226384 0.84 CHRNB2 (0.34) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2
SCHEMBL7224694 0.83 SLC6A3 (0.33) SLC6A3SLC6A4CHRNB2CHRNA4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed