SCHEMBL7224848

SCHEMBL7224848

COc1ccn2c(Br)cnc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 4/20 0.43
GABRB3 P28472 4/20 0.43
GABRA1 P14867 3/20 0.43
GABRA3 P34903 3/20 0.43
KDM4E B2RXH2 2/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KDR P35968 2/20 0.35
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GPR139 Q6DWJ6 2/20 0.32
GABRA5 P31644 1/20 0.31
PLA2G7 Q13093 1/20 0.31
PDE10A Q9Y233 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6217150 0.76 SMN1; SMN2 (0.33) GABRG2GABRB3GABRA1GABRA3KDM4E
SCHEMBL6216575 0.76 TDP1 (0.33) GABRG2GABRB3GABRA1GABRA3KDM4E
SCHEMBL7225436 0.73 MAPK1 (0.41) KDM4ERAB9ANPC1ALDH1A1KDR
SCHEMBL6217979 0.72 GABRA1 (0.34) GABRG2GABRB3GABRA1GABRA3
SCHEMBL31728622 0.71 ADORA3 (0.42) GABRG2GABRB3GABRA1GABRA3KDM4E
SCHEMBL5771903 0.70 GABRA1 (0.47) GABRG2GABRB3GABRA1GABRA3GABRA5
SCHEMBL6221519 0.70 GABRA1 (0.47) GABRG2GABRB3GABRA1GABRA3GABRA5
SCHEMBL31208206 0.69 TGFBR1 (0.52) GABRA1KDM4ERAB9AALDH1A1MAPT
SCHEMBL6219080 0.69 GABRA1 (0.36) GABRG2GABRB3GABRA1GABRA3ALDH1A1
SCHEMBL6221427 0.69 GABRA1 (0.34) GABRG2GABRB3GABRA1GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6642229-B2 Treatment of adverse neurological conditions MERCK SHARP & DOHME LTD. 2003-11-04 US disclosed