SCHEMBL7233270

SCHEMBL7233270

COc1ccccc1-c1ncc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.48
HDAC4 P56524 3/20 0.48
HDAC1 Q13547 3/20 0.48
HDAC7 Q8WUI4 3/20 0.48
HDAC2 Q92769 3/20 0.48
HDAC10 Q969S8 3/20 0.48
HDAC11 Q96DB2 3/20 0.48
HDAC8 Q9BY41 3/20 0.48
HDAC6 Q9UBN7 3/20 0.48
HDAC9 Q9UKV0 3/20 0.48
HDAC5 Q9UQL6 3/20 0.48
CHRNA7 P36544 1/20 0.43
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
USP30 Q70CQ3 1/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231070 0.88 SSTR4 (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7226023 0.87 USP30 (0.41) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7225952 0.87 MAPK14 (0.45) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7234311 0.86 USP30 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7075331 0.86 USP30 (0.39) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7225473 0.85 MAPK11 (0.42) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7233186 0.85 USP30 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL7230337 0.85 MAPK11 (0.49) HDAC1CHRNA7HTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL7077995 0.85 USP30 (0.39) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7224115 0.84 MAPK11 (0.43) CHRNA7HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed